PDB entry 3dk7
View 3dk7 on RCSB PDB site
Description: Crystal structure of mutant ABL kinase domain in complex with small molecule fragment
Class: transferase
Keywords: DRUG DISCOVERY, ABL KINASE, FRAGMENT BASED, Alternative splicing, ATP-binding, Cell adhesion, Chromosomal rearrangement, Cytoplasm, Cytoskeleton, Kinase, Lipoprotein, Magnesium, Manganese, Metal-binding, Myristate, Nucleotide-binding, Nucleus, Phosphoprotein, Proto-oncogene, SH2 domain, SH3 domain, Transferase
Deposited on
2008-06-24, released
2008-07-29
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2.01 Å
R-factor: 0.216
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene tyrosine-protein kinase ABL1
Species: Mus musculus [TaxId:10090]
Gene: Abl1, Abl
Database cross-references and differences (RAF-indexed):
- Uniprot P00520 (3-End)
- engineered (85)
- engineered (215)
Domains in SCOPe 2.02: d3dk7a_ - Chain 'B':
Compound: Proto-oncogene tyrosine-protein kinase ABL1
Species: Mus musculus [TaxId:10090]
Gene: Abl1, Abl
Database cross-references and differences (RAF-indexed):
- Uniprot P00520 (3-275)
- engineered (85)
- engineered (215)
Domains in SCOPe 2.02: d3dk7b_ - Heterogens: SO4, SX7, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3dk7A (A:)
gsldkwemertditmkhklgggqygevyegvwkkysltvavktlkedtmeveeflkeaav
mkeikhpnlvqllgvctreppfyiiiefmtygnlldylrecnrqevsavvllymatqiss
ameylekknfihrdlaarnclvgenhlvkvadfglsrlmtgdtytahagakfpikwtape
slaynkfsiksdvwafgvllweiatygmspypgidpsqvyellekdyrmerpegcpekvy
elmracwqwnpsdrpsfaeihqafetmfqessisdeg
Sequence, based on observed residues (ATOM records): (download)
>3dk7A (A:)
dkwemertditmkhklgggqygevyegvwkkysltvavktlkeveeflkeaavmkeikhp
nlvqllgvctreppfyiiiefmtygnlldylrecnrqevsavvllymatqissameylek
knfihrdlaarnclvgenhlvkvadfglsrlmtgdtytahagakfpikwtapeslaynkf
siksdvwafgvllweiatygmspypgidpsqvyellekdyrmerpegcpekvyelmracw
qwnpsdrpsfaeihqafetmfqessi
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3dk7B (B:)
gsldkwemertditmkhklgggqygevyegvwkkysltvavktlkedtmeveeflkeaav
mkeikhpnlvqllgvctreppfyiiiefmtygnlldylrecnrqevsavvllymatqiss
ameylekknfihrdlaarnclvgenhlvkvadfglsrlmtgdtytahagakfpikwtape
slaynkfsiksdvwafgvllweiatygmspypgidpsqvyellekdyrmerpegcpekvy
elmracwqwnpsdrpsfaeihqafetmfqessisdeg
Sequence, based on observed residues (ATOM records): (download)
>3dk7B (B:)
dkwemertditmkhklgggqygevyegvwkkysltvavktlmeveeflkeaavmkeikhp
nlvqllgvctreppfyiiiefmtygnlldylrecnrqevsavvllymatqissameylek
knfihrdlaarnclvgenhlvkvadfglsrlmtgdtytahagakfpikwtapeslaynkf
siksdvwafgvllweiatygmspypgidpsqvyellekdyrmerpegcpekvyelmracw
qwnpsdrpsfaeihqafetmfqessisde