PDB entry 3dj5
View 3dj5 on RCSB PDB site
Description: Crystal structure of the mouse Aurora-A catalytic domain (Asn186->Gly, Lys240->Arg, Met302->Leu) in complex with Compound 290.
Class: Transferase
Keywords: Aurora A, small-molecule inhibitor, fragment-based drug discovery, Kinase, Transferase
Deposited on
2008-06-22, released
2009-05-05
The last revision prior to the SCOPe 2.07 freeze date was dated
2009-05-05, with a file datestamp of
2009-05-01.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.21
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine kinase 6
Species: Mus musculus [TaxId:10090]
Gene: Aurka, Stk6
Database cross-references and differences (RAF-indexed):
- Uniprot Q8C3H8
- engineered (53)
- engineered (107)
- engineered (169)
Domains in SCOPe 2.07: d3dj5a_ - Heterogens: AK5, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3dj5A (A:)
gplgskrqwtledfdigrplgkgkfgnvylarerqskfilalkvlfktqlekagvehqlr
reveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklsrfdeqrtatyite
lanalsychskrvihrdikpenlllgsngelkiadfgwsvhapssrrttlcgtldylppe
miegrmhdekvdlwslgvlcyeflvgmppfeahtyqetyrrisrveftfpdfvtegardl
isrllkhnasqrltlaevlehpwikansskps
Sequence, based on observed residues (ATOM records): (download)
>3dj5A (A:)
wtledfdigrplgkgkfgnvylarerqskfilalkvlfktqlekagvehqlrreveiqsh
lrhpnilrlygyfhdatrvylileyaplgtvyrelqklsrfdeqrtatyitelanalsyc
hskrvihrdikpenlllgsngelkiadfgwttlcgtldylppemiegrmhdekvdlwslg
vlcyeflvgmppfeahtyqetyrrisrveftfpdfvtegardlisrllkhnasqrltlae
vlehpwikanss