PDB entry 3daj
View 3daj on RCSB PDB site
Description: Crystal structure of Aurora A complexed with an inhibitor discovered through site-directed dynamic tethering
Class: transferase
Keywords: Protein-small molecule inhibitor complex, Kinase, TRANSFERASE
Deposited on
2008-05-29, released
2008-07-08
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.253
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine kinase 6
Species: Mus musculus [TaxId:10090]
Gene: Aurka, Stk6
Database cross-references and differences (RAF-indexed):
- Uniprot Q8C3H8
- engineered (53)
- engineered (107)
Domains in SCOPe 2.01: d3daja_ - Heterogens: FXG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3dajA (A:)
gplgskrqwtledfdigrplgkgkfgnvylarerqskfilalkvlfktqlekagvehqlr
reveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklsrfdeqrtatyite
lanalsychskrvihrdikpenlllgsngelkiadfgwsvhapssrrdtlcgtldylppe
miegrmhdekvdlwslgvlcyeflvgmppfeahtyqetyrrisrveftfpdfvtegardl
isrllkhnasqrltlaevlehpwikansskps
Sequence, based on observed residues (ATOM records): (download)
>3dajA (A:)
qwtledfdigrplgkgkfgnvylarerqskfilalkvlfktqlekagvehqlrreveiqs
hlrhpnilrlygyfhdatrvylileyaplgtvyrelqklsrfdeqrtatyitelanalsy
chskrvihrdikpenlllgsngelkiadfgwstldylppemihdekvdlwslgvlcyefl
vgmppfeahtyqetyrrisrveftfpdfvtegardlisrllkhnasqrltlaevlehpwi
kanss