PDB entry 3d2i
View 3d2i on RCSB PDB site
Description: Crystal structure of mouse Aurora A (Asn186->Gly, Lys240->Arg, Met302->Leu) in complex with 1-{5-[2-(1-methyl-1H-pyrazolo[4,3-d]pyrimidin-7-ylamino)-ethyl]-thiazol-2-yl}-3-(3-trifluoromethyl-phenyl)-urea
Class: Transferase
Keywords: Aurora A, small-molecule inhibitor, Kinase, Transferase
Deposited on
2008-05-08, released
2009-05-12
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-05-12, with a file datestamp of
2009-05-08.
Experiment type: XRAY
Resolution: 2.9 Å
R-factor: 0.245
AEROSPACI score: 0.22
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine kinase 6
Species: Mus musculus [TaxId:10090]
Gene: Aurka, Stk6
Database cross-references and differences (RAF-indexed):
- Uniprot Q8C3H8
- engineered (53)
- engineered (107)
Domains in SCOPe 2.06: d3d2ia_ - Heterogens: AK3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3d2iA (A:)
gplgskrqwtledfdigrplgkgkfgnvylarerqskfilalkvlfktqlekagvehqlr
reveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklsrfdeqrtatyite
lanalsychskrvihrdikpenlllgsngelkiadfgwsvhapssrrttlcgtldylppe
miegrmhdekvdlwslgvlcyeflvgmppfeahtyqetyrrisrveftfpdfvtegardl
isrllkhnasqrltlaevlehpwikansskps
Sequence, based on observed residues (ATOM records): (download)
>3d2iA (A:)
qwtledfdigrplgkgkfgnvylarerqskfilalkvlfktqlekagvehqlrreveiqs
hlrhpnilrlygyfhdatrvylileyaplgtvyrelqklsrfdeqrtatyitelanalsy
chskrvihrdikpenlllgsngelkiadfgwsvhapcgtldylppemiegrmhdekvdlw
slgvlcyeflvgmppfeahtyqetyrrisrveftfpdfvtegardlisrllkhnasqrlt
laevlehpwikanss