PDB entry 3cjg

View 3cjg on RCSB PDB site
Description: Crystal structure of VEGFR2 in complex with a 3,4,5-trimethoxy aniline containing pyrimidine
Class: transferase
Keywords: Vascular endothelial growth factor receptor 2. vegfr-2, kinase insert domain receptor, protein-tyrosine kinase receptor flk-1, Angiogenesis, ATP-binding, Developmental protein, Differentiation, Glycoprotein, Host-virus interaction, Immunoglobulin domain, Membrane, Nucleotide-binding, Phosphoprotein, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on 2008-03-12, released 2008-10-07
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-10-25, with a file datestamp of 2017-10-20.
Experiment type: XRAY
Resolution: 2.25 Å
R-factor: N/A
AEROSPACI score: 0.25 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Vascular endothelial growth factor receptor 2
    Species: HOMO SAPIENS
    Gene: KDR, FLK1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P35968 (Start-133)
      • see remark 999 (29)
    • Uniprot P35968 (134-308)
    Domains in SCOPe 2.08: d3cjga_
  • Heterogens: SO4, KIM, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3cjgA (A:)
    mdpdelpldehcerlpydaskwefprdrlnlgkplgrgafgqvieadafgidktatcrtv
    avkmlkegathsehralmselkilihighhlnvvnllgactkpggplmvivefckfgnls
    tylrskrnefvpykdlykdfltlehlicysfqvakgmeflasrkcihrdlaarnillsek
    nvvkicdfglardiykdpdyvrkgdarlplkwmapetifdrvytiqsdvwsfgvllweif
    slgaspypgvkideefcrrlkegtrmrapdyttpemyqtmldcwhgepsqrptfselveh
    lgnllqana
    

    Sequence, based on observed residues (ATOM records): (download)
    >3cjgA (A:)
    hcerlpydaskwefprdrlnlgkplgrgqvieadafgidktatcrtvavkmlkegathse
    hralmselkilihighhlnvvnllgactkpggplmvivefckfgnlstylrskrnefvpy
    kdlykdfltlehlicysfqvakgmeflasrkcihrdlaarnillseknvvkicdfglard
    iplkwmapetifdrvytiqsdvwsfgvllweifslgaspypgvkideefcrrlkegtrmr
    apdyttpemyqtmldcwhgepsqrptfselvehlgnllqana