PDB entry 3cd8
View 3cd8 on RCSB PDB site
Description: X-ray Structure of c-Met with triazolopyridazine Inhibitor.
Class: transferase
Keywords: c-Met, Kinase, Triazolopyridazine, ATP-binding, Glycoprotein, Membrane, Nucleotide-binding, Phosphoprotein, Proto-oncogene, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2008-02-26, released
2008-04-29
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.236
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d3cd8a_ - Heterogens: L5G, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3cd8A (A:)
mqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkih
cavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlr
nfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfgla
rdmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypd
vntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig
ehyvhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3cd8A (A:)
dlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlkihcavkslnrigevs
qfltegiimkdfshpnvlsllgicsplvvlpymkhgdlrnfirnethnptvkdligfglq
vakgmkylaskkfvhrdlaarncmldekftvkvadfglardmydkeyysvhktgaklpvk
wmaleslqtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeyc
pdplyevmlkcwhpkaemrpsfselvsrisaifstfig