PDB entry 3c4f
View 3c4f on RCSB PDB site
Description: FGFR TYROSINE KINASE DOMAIN IN COMPLEX WITH 3-(3-methoxybenzyl)-7-azaindole
Class: transferase
Keywords: FIBROBLAST GROWTH FACTOR RECEPTOR, TYROSINE KINASE DOMAIN, RECEPTOR TYROSINE KINASE, FGFR1, FGFR, Alternative splicing, ATP-binding, Chromosomal rearrangement, Disease mutation, Dwarfism, Glycoprotein, Heparin-binding, Immunoglobulin domain, Kallmann syndrome, Membrane, Nucleotide-binding, Phosphoprotein, Polymorphism, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2008-01-29, released
2008-02-26
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 2.07 Å
R-factor: 0.213
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Basic fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, FGFBR, FLG, FLT2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3c4fa_ - Chain 'B':
Compound: Basic fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, FGFBR, FLG, FLT2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3c4fb_ - Heterogens: C4F, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3c4fA (A:)
elpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksdatek
dlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppgley
cynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfg
lardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypg
vpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsn
qe
Sequence, based on observed residues (ATOM records): (download)
>3c4fA (A:)
elpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksdatek
dlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppeeql
sskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfglardihhidyyk
kttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelfkllke
ghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsnqe
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3c4fB (B:)
elpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksdatek
dlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppgley
cynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfg
lardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypg
vpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsn
qe
Sequence, based on observed residues (ATOM records): (download)
>3c4fB (B:)
elpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksdatek
dlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppeeql
sskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfglardihhidyyk
kttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelfkllke
ghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsnqe