PDB entry 3bu5
View 3bu5 on RCSB PDB site
Description: Crystal structure of the insulin receptor kinase in complex with IRS2 KRLB peptide and ATP
Class: transferase
Keywords: IRK, KRLB, IRS2, ATP, insulin receptor, peptide, substrate, Alternative splicing, ATP-binding, Carbohydrate metabolism, Cleavage on pair of basic residues, Diabetes mellitus, Disease mutation, Glycoprotein, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Polymorphism, Transferase, Transmembrane, Tyrosine-protein kinase, Transducer
Deposited on
2007-12-31, released
2008-02-19
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.196
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: insulin receptor subunit beta
Species: Homo sapiens [TaxId:9606]
Gene: INSR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3bu5a_ - Chain 'B':
Compound: Insulin receptor substrate 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: MG, ATP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3bu5A (A:)
vfpssvyvpdewevsrekitllrelgqgsfgmvyegnardiikgeaetrvavktvnesas
lrerieflneasvmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaen
npgrppptlqemiqmaaeiadgmaylnakkfvhrdlaarncmvahdftvkigdfgmtrdi
yetdyyrkggkgllpvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsneq
vlkfvmdggyldqpdncpervtdlmrmcwqfnpnmrptfleivnllkddlhpsfpevsff
hseenk
Sequence, based on observed residues (ATOM records): (download)
>3bu5A (A:)
dewevsrekitllrelgqgmvyegnardiikgeaetrvavktvnesaslrerieflneas
vmkgftchhvvrllgvvskgqptlvvmelmahgdlksylrslrpeaennpgrppptlqem
iqmaaeiadgmaylnakkfvhrdlaarncmvahdftvkigdfgmtrdiyetdyyrkggkg
llpvrwmapeslkdgvfttssdmwsfgvvlweitslaeqpyqglsneqvlkfvmdggyld
qpdncpervtdlmrmcwqfnpnmrptfleivnllkddlhpsfpevsffhseenk
- Chain 'B':
No sequence available.