PDB entry 3bqr

View 3bqr on RCSB PDB site
Description: Crystal structure of human death associated protein kinase 3 (DAPK3) in complex with an imidazo-pyridazine ligand
Class: transferase
Keywords: Death Associated Kinase, DAPK3, ZIP kinase, ZIPK, DAP kinase 3, DAP like kinase, Dlk, Structural Genomics Consortium, SGC, Apoptosis, ATP-binding, Chromatin regulator, Nucleotide-binding, Nucleus, Serine/threonine-protein kinase, Transferase
Deposited on 2007-12-20, released 2008-02-26
The last revision prior to the SCOPe 2.06 freeze date was dated 2011-07-13, with a file datestamp of 2011-05-08.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: 0.181
AEROSPACI score: 0.54 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: death-associated protein kinase 3
    Species: Homo sapiens [TaxId:9606]
    Gene: DAPK3, ZIPK
    Database cross-references and differences (RAF-indexed):
    • Uniprot O43293 (2-End)
      • expression tag (0-1)
    Domains in SCOPe 2.06: d3bqra1, d3bqra2
  • Heterogens: 4RB, PGO, GOL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3bqrA (A:)
    smvedhyemgeelgsgqfaivrkcrqkgtgkeyaakfikkrrlsssrrgvsreeierevn
    ilreirhpniitlhdifenktdvvlilelvsggelfdflaekesltedeatqflkqildg
    vhylhskriahfdlkpenimlldknvpnpriklidfgiahkieagnefknifgtpefvap
    eivnyeplgleadmwsigvityillsgaspflgetkqetltnisavnydfdeeyfsntse
    lakdfirrllvkdpkrrmtiaqslehswikairrrnvrgedsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >3bqrA (A:)
    smvedhyemgeelgsgqfaivrkcrqkgtgkeyaakfikkrrlsssrrgvsreeierevn
    ilreirhpniitlhdifenktdvvlilelvsggelfdflaekesltedeatqflkqildg
    vhylhskriahfdlkpenimlldknvpnpriklidfgiahkieagnnifgtpefvapeiv
    nyeplgleadmwsigvityillsgaspflgetkqetltnisavnydfdeeyfsntselak
    dfirrllvkdpkrrmtiaqslehswikairrrnvr