PDB entry 3bea
View 3bea on RCSB PDB site
Description: cFMS tyrosine kinase (tie2 KID) in complex with a pyrimidinopyridone inhibitor
Class: transferase
Keywords: Kinase domain, inhibitor, transferase, juxtamembrane domain, ATP-binding, Glycoprotein, Immunoglobulin domain, Nucleotide-binding, Phosphoprotein, Polymorphism, Proto-oncogene, Receptor, Transmembrane, Tyrosine-protein kinase
Deposited on
2007-11-16, released
2008-07-15
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.02 Å
R-factor: 0.193
AEROSPACI score: 0.44
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Macrophage colony-stimulating factor 1 receptor
Species: HOMO SAPIENS
Gene: CSF1R, FMS
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3beaa_ - Heterogens: SO4, IXH, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3beaA (A:)
gvdykykqkpkyqvrwkiiesyegnsytfidptqlpynekwefprnnlqfgktlgagafg
kvveatafglgkedavlkvavkmlkstahadekealmselkimshlgqhenivnllgact
hggpvlviteyccygdllnflrrksrvletdpafaianstlstrdllhfssqvaqgmafl
askncihrdvaarnvlltnghvakigdfglardimndsnyivkgnarlpvkwmapesifd
cvytvqsdvwsygillweifslglnpypgilvnskfyklvkdgyqmaqpafapkniysim
qacwalepthrptfqqicsflqeqaqedrrerd
Sequence, based on observed residues (ATOM records): (download)
>3beaA (A:)
qvrwkiiesyegnsytfidptqlpynekwefprnnlqfgktlgagafgkvveatafglgk
edavlkvavkmlkstahadekealmselkimshlgqhenivnllgacthggpvlviteyc
cygdllnflrrksrvlstlstrdllhfssqvaqgmaflaskncihrdvaarnvlltnghv
akigdfglardimndsnyivkgnarlpvkwmapesifdcvytvqsdvwsygillweifsl
glnpypgilvnskfyklvkdgyqmaqpafapkniysimqacwalepthrptfqqicsflq
eqaqedrrer