PDB entry 3ara
View 3ara on RCSB PDB site
Description: Discovery of Novel Uracil Derivatives as Potent Human dUTPase Inhibitors
Class: Hydrolase/Hydrolase inhibitor
Keywords: Hydrolase, Magnesium Binding, Hydrolase-Hydrolase inhibitor complex
Deposited on
2010-11-25, released
2010-12-08
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-11, with a file datestamp of
2017-10-06.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: N/A
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: deoxyuridine 5'-triphosphate nucleotidohydrolase
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3araa_ - Chain 'B':
Compound: deoxyuridine 5'-triphosphate nucleotidohydrolase
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3arab_ - Chain 'C':
Compound: deoxyuridine 5'-triphosphate nucleotidohydrolase
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3arac_ - Heterogens: MKH, MG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3araA (A:)
mpcseetpaispskrarpaevggmqlrfarlsehataptrgsaraagydlysaydytipp
mekavvktdiqialpsgcygrvaprsglaakhfidvgagvidedyrgnvgvvlfnfgkek
fevkkgdriaqlicerifypeieevqalddtergsggfgstgkn
Sequence, based on observed residues (ATOM records): (download)
>3araA (A:)
mqlrfarlsehataptrgsaraagydlysaydytippmekavvktdiqialpsgcygrva
prsglaakhfidvgagvidedyrgnvgvvlfnfgkekfevkkgdriaqlicerifypeie
evqal
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3araB (B:)
mpcseetpaispskrarpaevggmqlrfarlsehataptrgsaraagydlysaydytipp
mekavvktdiqialpsgcygrvaprsglaakhfidvgagvidedyrgnvgvvlfnfgkek
fevkkgdriaqlicerifypeieevqalddtergsggfgstgkn
Sequence, based on observed residues (ATOM records): (download)
>3araB (B:)
mqlrfarlsehataptrgsaraagydlysaydytippmekavvktdiqialpsgcygrva
prsglaakhfidvgagvidedyrgnvgvvlfnfgkekfevkkgdriaqlicerifypeie
evqal
- Chain 'C':
Sequence, based on SEQRES records: (download)
>3araC (C:)
mpcseetpaispskrarpaevggmqlrfarlsehataptrgsaraagydlysaydytipp
mekavvktdiqialpsgcygrvaprsglaakhfidvgagvidedyrgnvgvvlfnfgkek
fevkkgdriaqlicerifypeieevqalddtergsggfgstgkn
Sequence, based on observed residues (ATOM records): (download)
>3araC (C:)
mqlrfarlsehataptrgsaraagydlysaydytippmekavvktdiqialpsgcygrva
prsglaakhfidvgagvidedyrgnvgvvlfnfgkekfevkkgdriaqlicerifypeie
evqal