PDB entry 2zv2
View 2zv2 on RCSB PDB site
Description: Crystal structure of human calcium/calmodulin-dependent protein kinase kinase 2, beta, CaMKK2 kinase domain in complex with STO-609
Class: transferase/transferase inhibitor
Keywords: calcium/calmodulin-dependent protein kinase kinase 2, beta, STO-609, CaMKK2, E.C.2.7.11.17, Phosphorylation, AMPKK, metabolism, ATP-binding, kinase, Calmodulin-binding, Nucleotide-binding, Phosphoprotein, Serine/threonine-protein kinase, Transferase, Structural Genomics, NPPSFA, National Project on Protein Structural and Functional Analyses, RIKEN Structural Genomics/Proteomics Initiative, RSGI, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2008-10-31, released
2009-11-03
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-11-20, with a file datestamp of
2013-11-15.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.203
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Calcium/calmodulin-dependent protein kinase kinase 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2zv2a_ - Heterogens: 609, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2zv2A (A:)
gssgssgdcvqlnqytlkdeigkgsygvvklaynendntyyamkvlskkklirqagfprr
ppprgtrpapggciqprgpieqvyqeiailkkldhpnvvklvevlddpnedhlymvfelv
nqgpvmevptlkplsedqarfyfqdlikgieylhyqkiihrdikpsnllvgedghikiad
fgvsnefkgsdallsntvgtpafmapeslsetrkifsgkaldvwamgvtlycfvfgqcpf
mderimclhskiksqalefpdqpdiaedlkdlitrmldknpesrivvpeiklhpwvtr
Sequence, based on observed residues (ATOM records): (download)
>2zv2A (A:)
vqlnqytlkdeigkygvvklaynendntyyamkvlskkeqvyqeiailkkldhpnvvklv
evlddpnedhlymvfelvnqgpvmevptlkplsedqarfyfqdlikgieylhyqkiihrd
ikpsnllvgedghikiadfgvsnefkgsdallsntvgtpafmapeslsetrkifsgkald
vwamgvtlycfvfgqcpfmderimclhskiksqalefpdqpdiaedlkdlitrmldknpe
srivvpeiklhpwvtr