PDB entry 2ycr
View 2ycr on RCSB PDB site
Description: crystal structure of checkpoint kinase 2 in complex with inhibitor pv976
Class: transferase
Keywords: transferase, anticancer drug design
Deposited on
2011-03-16, released
2011-11-16
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-11-16, with a file datestamp of
2011-11-11.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.20206
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase chk2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2ycra_ - Heterogens: HCW, NO3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2ycrA (A:)
msvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsareadpal
nveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyf
yqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmrtlcgtp
tylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfi
pevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllseenestak
pqvlaqpstsrkrpregeaegae
Sequence, based on observed residues (ATOM records): (download)
>2ycrA (A:)
vypkalrdeyimsktlgsgevklaferktckkvaikiisknveteieilkklnhpciiki
knffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengiihrdl
kpenvllssqeedclikitdfghskilgetslmrtlcgtptylapevlvsvgtagynrav
dcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvkkllv
vdpkarftteealrhpwlqdedmkrkfqdllseenestakpq