PDB entry 2ycf

View 2ycf on RCSB PDB site
Description: crystal structure of checkpoint kinase 2 in complex with inhibitor pv1531
Class: transferase
Keywords: transferase, anticancer, anticancer drug design
Deposited on 2011-03-14, released 2011-11-16
The last revision prior to the SCOPe 2.08 freeze date was dated 2011-11-16, with a file datestamp of 2011-11-11.
Experiment type: XRAY
Resolution: 1.77 Å
R-factor: 0.19739
AEROSPACI score: 0.52 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: serine/threonine-protein kinase chk2
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d2ycfa_
  • Heterogens: YCF, MG, NO3, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >2ycfA (A:)
    msvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsareadpal
    nveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyf
    yqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmrtlcgtp
    tylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfi
    pevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllseenestal
    pqvlaqpstsrkrpregeaega
    

    Sequence, based on observed residues (ATOM records): (download)
    >2ycfA (A:)
    svypkalrdeyimsktlgsgacgevklaferktckkvaikiisknveteieilkklnhpc
    iikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengii
    hrdlkpenvllssqeedclikitdfghskilgetslmrtlcgtptylapevlvsvgtagy
    nravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvk
    kllvvdpkarftteealrhpwlqdedmkrkfqdllseenestalpq