PDB entry 2ycf
View 2ycf on RCSB PDB site
Description: crystal structure of checkpoint kinase 2 in complex with inhibitor pv1531
Class: transferase
Keywords: transferase, anticancer, anticancer drug design
Deposited on
2011-03-14, released
2011-11-16
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-11-16, with a file datestamp of
2011-11-11.
Experiment type: XRAY
Resolution: 1.77 Å
R-factor: 0.19739
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase chk2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2ycfa_ - Heterogens: YCF, MG, NO3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2ycfA (A:)
msvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsareadpal
nveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyf
yqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmrtlcgtp
tylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfi
pevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllseenestal
pqvlaqpstsrkrpregeaega
Sequence, based on observed residues (ATOM records): (download)
>2ycfA (A:)
svypkalrdeyimsktlgsgacgevklaferktckkvaikiisknveteieilkklnhpc
iikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengii
hrdlkpenvllssqeedclikitdfghskilgetslmrtlcgtptylapevlvsvgtagy
nravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvk
kllvvdpkarftteealrhpwlqdedmkrkfqdllseenestalpq