PDB entry 2xir

View 2xir on RCSB PDB site
Description: crystal structure of the vegfr2 kinase domain in complex with pf- 00337210 (n,2-dimethyl-6-(7-(2-morpholinoethoxy)quinolin-4-yloxy) benzofuran-3-carboxamide)
Deposited on 2010-06-30, released 2011-04-13
The last revision was dated 2019-05-08, with a file datestamp of 2019-05-03.
Experiment type: XRAY
Resolution: 1.5 Å
R-factor: N/A
AEROSPACI score: 0.48 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Vascular endothelial growth factor receptor 2
    Species: HOMO SAPIENS, synthetic [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
  • Heterogens: 00J, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >2xirA (A:)
    mdpdelpldehcerlpydaskwefprdrlklgkplgrgafgqvieadafgidktatcrtv
    avkmlkegathsehralmselkilihighhlnvvnllgactkpggplmvivefckfgnls
    tylrskrnefvpykvapedlykdfltlehlicysfqvakgmeflasrkcihrdlaarnil
    lseknvvkicdfglardiykdpdyvrkgdarlplkwmapetifdrvytiqsdvwsfgvll
    weifslgaspypgvkideefcrrlkegtrmrapdyttpemyqtmldcwhgepsqrptfse
    lvehlgnllqanaqqd
    

    Sequence, based on observed residues (ATOM records):
    >2xirA (A:)
    hcerlpydaskwefprdrlklgkplgrgafgqvieadafgidktatcrtvavkmlkegat
    hsehralmselkilihighhlnvvnllgactkpggplmvivefckfgnlstylrskrnef
    vpyykdfltlehlicysfqvakgmeflasrkcihrdlaarnillseknvvkicdfglard
    iykdpdyvrkgdarlplkwmapetifdrvytiqsdvwsfgvllweifslgaspypgvkid
    eefcrrlkegtrmrapdyttpemyqtmldcwhgepsqrptfselvehlgnllqana