PDB entry 2xgm

View 2xgm on RCSB PDB site
Description: substrate and product analogues as human o-glcnac transferase inhibitors.
Deposited on 2010-06-07, released 2010-08-25
The last revision was dated 2011-10-12, with a file datestamp of 2011-10-07.
Experiment type: XRAY
Resolution: 2.55 Å
R-factor: 0.268
AEROSPACI score: 0.23 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: xcogt
    Species: Xanthomonas campestris [TaxId:339]
    Database cross-references and differences (RAF-indexed):
  • Chain 'B':
    Compound: xcogt
    Species: Xanthomonas campestris [TaxId:339]
    Database cross-references and differences (RAF-indexed):
  • Heterogens: LXN, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >2xgmA (A:)
    mtadgprellqlraavrhrpqdfvawlmladaelgmgdttagemavqrglalhpghpeav
    arlgrvrwtqqrhaeaavllqqasdaapehpgialwlghaledagqaeaaaaaytrahql
    lpeepyitaqllnwrrrlcdwraldvlsaqvraavaqgvgavepfaflsedasaaeqlac
    artraqaiaasvrplaptrvrskgplrvgfvsngfgahptglltvalfealqrrqpdlqm
    hlfatsgddgstlrtrlaqastlhdvtalghlatakhirhhgidllfdlrgwggggrpev
    falrpapvqvnwlaypgtsgapwmdyvlgdafalppalepfysehvlrlqgafqpsdtsr
    vvaeppsrtqcglpeqgvvlccfnnsyklnpqsmarmlavlrevpdsvlwllsgpgeada
    rlrafahaqgvdaqrlvfmpklphpqylaryrhadlfldthpynahttasdalwtgcpvl
    ttpgetfaarvagslnhhlgldemnvaddaafvakavalasdpaaltalharvdvlrras
    gvfhmdgfaddfgallqalarrhgwlgi
    

    Sequence, based on observed residues (ATOM records):
    >2xgmA (A:)
    peavarlgrvrwtqqrhaeaavllqqasdaapehpgialwlghaledagqaeaaaaaytr
    ahqllpeepyitaqllnwrrrlcdwraldvlsaqvraavaqgvgavepfaflsedasaae
    qlacartraqaiaasvrplaptrvrskgplrvgfvsngfgahptglltvalfealqrrqp
    dlqmhlfatsgddgstlrtrlaqastlhdvtalghlatakhirhhgidllfdlrgwgggg
    rpevfalrpapvqvnwlaypgtsgapwmdyvlgdafalppalepfysehvlrlqgafqps
    dtsrvvaeppsrtqcglpeqgvvlccfnnsyklnpqsmarmlavlrevpdsvlwllsgpg
    eadarlrafahaqgvdaqrlvfmpklphpqylaryrhadlfldthpynahttasdalwtg
    cpvlttpgetfaarvagslnhhlgldemnvaddaafvakavalasdpaaltalharvdvl
    rrasgvfhmdgfaddfgallqalarrhgwlgi
    

  • Chain 'B':
    Sequence, based on SEQRES records:
    >2xgmB (B:)
    mtadgprellqlraavrhrpqdfvawlmladaelgmgdttagemavqrglalhpghpeav
    arlgrvrwtqqrhaeaavllqqasdaapehpgialwlghaledagqaeaaaaaytrahql
    lpeepyitaqllnwrrrlcdwraldvlsaqvraavaqgvgavepfaflsedasaaeqlac
    artraqaiaasvrplaptrvrskgplrvgfvsngfgahptglltvalfealqrrqpdlqm
    hlfatsgddgstlrtrlaqastlhdvtalghlatakhirhhgidllfdlrgwggggrpev
    falrpapvqvnwlaypgtsgapwmdyvlgdafalppalepfysehvlrlqgafqpsdtsr
    vvaeppsrtqcglpeqgvvlccfnnsyklnpqsmarmlavlrevpdsvlwllsgpgeada
    rlrafahaqgvdaqrlvfmpklphpqylaryrhadlfldthpynahttasdalwtgcpvl
    ttpgetfaarvagslnhhlgldemnvaddaafvakavalasdpaaltalharvdvlrras
    gvfhmdgfaddfgallqalarrhgwlgi
    

    Sequence, based on observed residues (ATOM records):
    >2xgmB (B:)
    lmladaelgmgdttagemavqrglalhpghpeavarlgrvrwtqqrhaeaavllqqasda
    apehpgialwlghaledagqaeaaaaaytrahqllpeepyitaqllnwrrrlcdwraldv
    lsaqvraavaqgvgavepfaflsedasaaeqlacartraqaiaasvrplaptrvrskgpl
    rvgfvsngfgahptglltvalfealqrrqpdlqmhlfatsgddgstlrtrlaqastlhdv
    talghlatakhirhhgidllfdlrgwggggrpevfalrpapvqvnwlaypgtsgapwmdy
    vlgdafalppalepfysehvlrlqgafqpsdtsrvvaeppsrtqcglpeqgvvlccfnns
    yklnpqsmarmlavlrevpdsvlwllsgpgeadarlrafahaqgvdaqrlvfmpklphpq
    ylaryrhadlfldthpynahttasdalwtgcpvlttpgetfaarvagslnhhlgldemnv
    addaafvakavalasdpaaltalharvdvlrrasgvfhmdgfaddfgallqalarrhgwl
    gi