PDB entry 2wxe

View 2wxe on RCSB PDB site
Description: the crystal structure of the murine class ia pi 3-kinase p110delta in complex with ic87114.
Deposited on 2009-11-09, released 2010-01-12
The last revision was dated 2010-02-02, with a file datestamp of 2010-01-29.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.24074
AEROSPACI score: 0.33 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta isoform
    Species: Mus musculus [TaxId:10090]
    Database cross-references and differences (RAF-indexed):
  • Heterogens: IC8, HOH

PDB Chain Sequences:
This PDB entry is not classified in SCOPe 2.08, so the chain sequences below are not included in the ASTRAL sequence sets.

  • Chain 'A':
    Sequence, based on SEQRES records:
    >2wxeA (A:)
    ggdrvkklinsqislligkglhefdslrdpevndfrtkmrqfceeaaahrqqlgwvewlq
    ysfplqlepsargwragllrvsnrallvnvkfegseesftfqvstkdmplalmacalrkk
    atvfrqplveqpeeyalqvngrheylygnyplchfqyicsclhsgltphltmvhsssila
    mrdeqsnpapqvqkprakpppipakkpssvslwsleqpfsieliegrkvnadermklvvq
    aglfhgnemlcktvsssevnvcsepvwkqrlefdisvcdlprmarlcfalyavvekakka
    rstkkkskkadcpiawanlmlfdykdqlktgerclymwpsvpdekgellnpagtvrgnpn
    tesaaalviylpevaphpvyfpalekilelgrhgergriteeeqlqlreilerrgsgely
    ehekdlvwkmrhevqehfpealarlllvtkwnkhedvaqmlyllcswpelpvlsalelld
    fsfpdcyvgsfaikslrkltddelfqyllqlvqvlkyesyldceltkfllgralanrkig
    hflfwhlrsemhvpsvalrfglimeaycrgsthhmkvlmkqgealsklkalndfvkvssq
    kttkpqtkemmhmcmrqetymealshlqspldpstlleevcveqctfmdskmkplwimys
    seeagsagnvgiifkngddlrqdmltlqmiqlmdvlwkqegldlrmtpygclptgdrtgl
    ievvlhsdtianiqlnksnmaataafnkdallnwlksknpgealdraieeftlscagycv
    atyvlgigdrhsdnimiresgqlfhidfghflgnfktkfginrervpfiltydfvhviqq
    gktnnsekferfrgyceraytilrrhgllflhlfalmraaglpelscskdiqylkdslal
    gkteeealkhfrvkfnealreswktkvnwlahnvskdnrq
    

    Sequence, based on observed residues (ATOM records):
    >2wxeA (A:)
    vkklinsqislligkglhefdslrdpevndfrtkmrqfceeaaahrqqlgwvewlqysfp
    lqlepnrallvnvkfegseesftfqvstkdmplalmacalrkkatvfrqqpeeyalqvng
    rheylygnyplchfqyicsclhsgltphltmvhsssilamrdeqsnlwsleqpfsielie
    grkvnamklvvqaglfhgnemlcktvsssevnvcsepvwkqrlefdisvcdlprmarlcf
    alyavvdcpiawanlmlfdykdqlktgerclymwpsvllnpagtvrgnpntesaaalviy
    lpevapvyfpalekilellreilerelyehekdlvwkmrhevqehfpealarlllvtkwn
    khedvaqmlyllcswpelpvlsalelldfsfpdcyvgsfaikslrkltddelfqyllqlv
    qvlkyesyldceltkfllgralanrkighflfwhlrsemhvpsvalrfglimeaycrgst
    hhmkvlmkqgealsklkalndfvkvssqkttkpqtkemmhmcmrqetymealshlqspld
    pstlleevcveqctfmdskmkplwimysseeagsagnvgiifkngddlrqdmltlqmiql
    mdvlwkqegldlrmtpygclptgdrtglievvlhsdtianiqlnksnmaataafnkdall
    nwlksknpgealdraieeftlscagycvatyvlgigdrhsdnimiresgqlfhidfghfl
    gnfrvpfiltydfvhviqqgktnnsekferfrgyceraytilrrhgllflhlfalmraag
    lpelscskdiqylkdslalgkteeealkhfrvkfnealresw