PDB entry 2wtd
View 2wtd on RCSB PDB site
Description: crystal structure of chk2 in complex with an inhibitor
Class: transferase
Keywords: transferase, kinase, cell cycle, li-fraumeni syndrome
Deposited on
2009-09-15, released
2009-12-29
The last revision prior to the SCOPe 2.08 freeze date was dated
2010-02-16, with a file datestamp of
2010-02-12.
Experiment type: XRAY
Resolution: 2.75 Å
R-factor: 0.194
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase chk2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- PDB 2WTD
- Uniprot O96017 (7-End)
Domains in SCOPe 2.08: d2wtda_ - Heterogens: ZZK, NO3, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2wtdA (A:)
gplgshmsvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsar
eadpalnveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkea
tcklyfyqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmr
tlcgtptylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqits
gkynfipevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllsee
nestalpqvlaqpstsrkrpregeaegae
Sequence, based on observed residues (ATOM records): (download)
>2wtdA (A:)
svypkalrdeyimsktlgsevklaferktckkvaikiiskpalnveteieilkklnhpci
ikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengiih
rdlkpenvllssqeedclikitdfghskiltslmrtlcgtptylapevlvsvgtagynra
vdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvkkll
vvdpkarftteealrhpwlqdedmkrkfqdllseenestalpqvl