PDB entry 2wtd

View 2wtd on RCSB PDB site
Description: crystal structure of chk2 in complex with an inhibitor
Class: transferase
Keywords: transferase, kinase, cell cycle, li-fraumeni syndrome
Deposited on 2009-09-15, released 2009-12-29
The last revision prior to the SCOPe 2.08 freeze date was dated 2010-02-16, with a file datestamp of 2010-02-12.
Experiment type: XRAY
Resolution: 2.75 Å
R-factor: 0.194
AEROSPACI score: 0.29 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: serine/threonine-protein kinase chk2
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
    • PDB 2WTD
    • Uniprot O96017 (7-End)
    Domains in SCOPe 2.08: d2wtda_
  • Heterogens: ZZK, NO3, EDO, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >2wtdA (A:)
    gplgshmsvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsar
    eadpalnveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkea
    tcklyfyqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmr
    tlcgtptylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqits
    gkynfipevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllsee
    nestalpqvlaqpstsrkrpregeaegae
    

    Sequence, based on observed residues (ATOM records): (download)
    >2wtdA (A:)
    svypkalrdeyimsktlgsevklaferktckkvaikiiskpalnveteieilkklnhpci
    ikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengiih
    rdlkpenvllssqeedclikitdfghskiltslmrtlcgtptylapevlvsvgtagynra
    vdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvkkll
    vvdpkarftteealrhpwlqdedmkrkfqdllseenestalpqvl