PDB entry 2waj
View 2waj on RCSB PDB site
Description: crystal structure of human jnk3 complexed with a 1-aryl-3,4-dihydroisoquinoline inhibitor
Class: transferase
Keywords: kinase, epilepsy, transferase, serine/threonine-protein kinase, ATP-binding, phosphoprotein, protein kinase, nucleotide-binding
Deposited on
2009-02-08, released
2009-03-31
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-07-13, with a file datestamp of
2011-06-02.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.187
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 10
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2waja_ - Heterogens: SNB, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2wajA (A:)
mskskvdnqfysvevgdstftvlkryqnlkpigsgaqgivcaaydavldrnvaikklsrp
fqnqthakrayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviq
meldhermsyllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartagtsf
mmtpyvvtryyrapevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieq
lgtpcpefmkklqptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardllsk
mlvidpakrisvddalqhpyinvwydpaeveapppqiydkqlderehtieewkeliykev
mnse
Sequence, based on observed residues (ATOM records): (download)
>2wajA (A:)
nqfysvevgdstftvlkryqnlkpigsggivcaaydavldrnvaikklsrpfqnqthakr
ayrelvlmkcvnhkniisllnvftpqktleefqdvylvmelmdanlcqviqmeldherms
yllyqmlcgikhlhsagiihrdlkpsnivvksdctlkildfglartsfmmtpyvvtryyr
apevilgmgykenvdiwsvgcimgemvrhkilfpgrdyidqwnkvieqlgtpcpefmkkl
qptvrnyvenrpkyagltfpklfpdslfpadsehnklkasqardllskmlvidpakrisv
ddalqhpyinvwydpaeveapppqdkqlderehtieewkeliykevmn