PDB entry 2vx3

View 2vx3 on RCSB PDB site
Description: Crystal structure of the human dual specificity tyrosine- phosphorylation-regulated kinase 1A
Class: transferase
Keywords: serine/threonine-protein kinase, minibrain homolog, nucleotide-binding, transferase, phosphoprotein, tyrosine-protein kinase, casp8, kinase
Deposited on 2008-06-30, released 2008-09-16
The last revision prior to the SCOPe 2.08 freeze date was dated 2013-06-26, with a file datestamp of 2013-06-21.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.186
AEROSPACI score: 0.38 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: dual specificity tyrosine-phosphorylation- regulated kinase 1a
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d2vx3a_
  • Chain 'B':
    Compound: dual specificity tyrosine-phosphorylation- regulated kinase 1a
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d2vx3b_
  • Chain 'C':
    Compound: dual specificity tyrosine-phosphorylation- regulated kinase 1a
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d2vx3c_
  • Chain 'D':
    Compound: dual specificity tyrosine-phosphorylation- regulated kinase 1a
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d2vx3d_
  • Heterogens: D15, CL, P6G, SO4, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >2vx3A (A:)
    mhhhhhhssgvdlgtenlyfqsmsshkkerkvyndgydddnydyivkngekwmdryeids
    ligkgsfgqvvkaydrveqewvaikiiknkkaflnqaqievrllelmnkhdtemkyyivh
    lkrhfmfrnhlclvfemlsynlydllrntnfrgvslnltrkfaqqmctallflatpelsi
    ihcdlkpenillcnpkrsaikivdfgsscqlgqriyqyiqsrfyrspevllgmpydlaid
    mwslgcilvemhtgeplfsganevdqmnkivevlgippahildqapkarkffeklpdgtw
    nlkktkdgkreykppgtrklhnilgvetggpggrragesghtvadylkfkdlilrmldyd
    pktriqpyyalqhsffkktade
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vx3A (A:)
    vyndgydddnydyivkngekwmdryeidsligkgsfgqvvkaydrveqewvaikiiknkk
    aflnqaqievrllelmnkhdtemkyyivhlkrhfmfrnhlclvfemlsynlydllrntnf
    rgvslnltrkfaqqmctallflatpelsiihcdlkpenillcnpkrsaikivdfgsscql
    gqriyqyiqsrfyrspevllgmpydlaidmwslgcilvemhtgeplfsganevdqmnkiv
    evlgippahildqapkarkffeklpdgtwnlkktkdgkreykppgtrklhnilgvetggp
    ggrragesghtvadylkfkdlilrmldydpktriqpyyalqhsffkk
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >2vx3B (B:)
    mhhhhhhssgvdlgtenlyfqsmsshkkerkvyndgydddnydyivkngekwmdryeids
    ligkgsfgqvvkaydrveqewvaikiiknkkaflnqaqievrllelmnkhdtemkyyivh
    lkrhfmfrnhlclvfemlsynlydllrntnfrgvslnltrkfaqqmctallflatpelsi
    ihcdlkpenillcnpkrsaikivdfgsscqlgqriyqyiqsrfyrspevllgmpydlaid
    mwslgcilvemhtgeplfsganevdqmnkivevlgippahildqapkarkffeklpdgtw
    nlkktkdgkreykppgtrklhnilgvetggpggrragesghtvadylkfkdlilrmldyd
    pktriqpyyalqhsffkktade
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vx3B (B:)
    vyndgydddnydyivkngekwmdryeidsligkgsfgqvvkaydrveqewvaikiiknkk
    aflnqaqievrllelmnkhdtemkyyivhlkrhfmfrnhlclvfemlsynlydllrntnf
    rgvslnltrkfaqqmctallflatpelsiihcdlkpenillcnpkrsaikivdfgsscql
    gqriyqyiqsrfyrspevllgmpydlaidmwslgcilvemhtgeplfsganevdqmnkiv
    evlgippahildqapkarkffeklpdgtwnlkkteykppgtrklhnilgvetggpggrra
    gesghtvadylkfkdlilrmldydpktriqpyyalqhsffk
    

  • Chain 'C':
    Sequence, based on SEQRES records: (download)
    >2vx3C (C:)
    mhhhhhhssgvdlgtenlyfqsmsshkkerkvyndgydddnydyivkngekwmdryeids
    ligkgsfgqvvkaydrveqewvaikiiknkkaflnqaqievrllelmnkhdtemkyyivh
    lkrhfmfrnhlclvfemlsynlydllrntnfrgvslnltrkfaqqmctallflatpelsi
    ihcdlkpenillcnpkrsaikivdfgsscqlgqriyqyiqsrfyrspevllgmpydlaid
    mwslgcilvemhtgeplfsganevdqmnkivevlgippahildqapkarkffeklpdgtw
    nlkktkdgkreykppgtrklhnilgvetggpggrragesghtvadylkfkdlilrmldyd
    pktriqpyyalqhsffkktade
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vx3C (C:)
    vyndgydddnydyivkngekwmdryeidsligkgsfgqvvkaydrveqewvaikiiknkk
    aflnqaqievrllelmnkhmkyyivhlkrhfmfrnhlclvfemlsynlydllrntnfrgv
    slnltrkfaqqmctallflatpelsiihcdlkpenillcnpkrsaikivdfgsscqlgqr
    iyqyiqsrfyrspevllgmpydlaidmwslgcilvemhtgeplfsganevdqmnkivevl
    gippahildqapkarkffeklpdgtwnlkktkdkreykppgtrklhnilgvetggpggrr
    sghtvadylkfkdlilrmldydpktriqpyyalqhsffk
    

  • Chain 'D':
    Sequence, based on SEQRES records: (download)
    >2vx3D (D:)
    mhhhhhhssgvdlgtenlyfqsmsshkkerkvyndgydddnydyivkngekwmdryeids
    ligkgsfgqvvkaydrveqewvaikiiknkkaflnqaqievrllelmnkhdtemkyyivh
    lkrhfmfrnhlclvfemlsynlydllrntnfrgvslnltrkfaqqmctallflatpelsi
    ihcdlkpenillcnpkrsaikivdfgsscqlgqriyqyiqsrfyrspevllgmpydlaid
    mwslgcilvemhtgeplfsganevdqmnkivevlgippahildqapkarkffeklpdgtw
    nlkktkdgkreykppgtrklhnilgvetggpggrragesghtvadylkfkdlilrmldyd
    pktriqpyyalqhsffkktade
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vx3D (D:)
    vyndgydddnydyivkngekwmdryeidsligkgsfgqvvkaydrveqewvaikiiknkk
    aflnqaqievrllelmnkhdtemkyyivhlkrhfmfrnhlclvfemlsynlydllrntnf
    rgvslnltrkfaqqmctallflatpelsiihcdlkpenillcnpkrsaikivdfgsscql
    gqriyqyiqsrfyrspevllgmpydlaidmwslgcilvemhtgeplfsganevdqmnkiv
    evlgippahildqapkarkffeklpdgtwnlkktkreykppgtrklhnilgvetggpggr
    ragesghtvadylkfkdlilrmldydpktriqpyyalqhsffk