PDB entry 2vwm
View 2vwm on RCSB PDB site
Description: aminopyrrolidine factor xa inhibitor
Class: blood clotting
Keywords: hydrolase, cation, plasma, calcium, zymogen, protease, inhibitor, polymorphism, glycoprotein, gamma-carboxyglutamic acid, blood clotting, coagulation factor, hydroxylation, serine protease, egf-like domain, cleavage on pair of basic residues
Deposited on
2008-06-26, released
2009-07-07
The last revision prior to the SCOPe 2.03 freeze date was dated
2009-07-07, with a file datestamp of
2009-07-02.
Experiment type: XRAY
Resolution: 1.96 Å
R-factor: 0.204
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: activated factor xa heavy chain
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P00742 (71-128)
- engineered mutation (137)
Domains in SCOPe 2.03: d2vwma_ - Chain 'B':
Compound: activated factor xa heavy chain
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P00742 (71-128)
- engineered mutation (137)
Domains in SCOPe 2.03: d2vwmb_ - Chain 'K':
Compound: factor x light chain
Species: Homo sapiens [TaxId:9606]
Domains in SCOPe 2.03: d2vwmk_ - Chain 'L':
Compound: factor x light chain
Species: Homo sapiens [TaxId:9606]
Domains in SCOPe 2.03: d2vwml_ - Heterogens: LZI, NA, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2vwmA (A:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlm
tqktgivsgfgrthekgeqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqeda
cqgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmktrglpka
k
Sequence, based on observed residues (ATOM records): (download)
>2vwmA (A:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlmt
qktgivsgfgrthekgeqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqedac
qgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2vwmB (B:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgdrnte
qeeggeavhevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlm
tqktgivsgfgrthekgeqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqeda
cqgdsggphvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmktrglpka
k
Sequence, based on observed residues (ATOM records): (download)
>2vwmB (B:)
ivggqeckdgecpwqallineenegfcggtilsefyiltaahclyqakrfkvrvgggeav
hevevvikhnrftketydfdiavlrlktpitfrmnvapaclperdwaestlmtqktgivs
gfgrthekgeqstrlkmlevpyvdrnscklsssfiitqnmfcagydtkqedacqgdsggp
hvtrfkdtyfvtgivswgegcarkgkygiytkvtaflkwidrsmk
- Chain 'K':
Sequence, based on SEQRES records: (download)
>2vwmK (K:)
rklcsldngdcdqfcheeqnsvvcscargytladngkaciptgpypcgkqtlerr
Sequence, based on observed residues (ATOM records): (download)
>2vwmK (K:)
rklcsldngdcdqfcheeqnsvvcscargytladngkaciptgpypcgkqtler
- Chain 'L':
Sequence, based on SEQRES records: (download)
>2vwmL (L:)
rklcsldngdcdqfcheeqnsvvcscargytladngkaciptgpypcgkqtlerr
Sequence, based on observed residues (ATOM records): (download)
>2vwmL (L:)
rklcsldngdcdqfcheeqnsvvcscargytladngkaciptgpypcgkqtl