PDB entry 2vt4

View 2vt4 on RCSB PDB site
Description: turkey beta1 adrenergic receptor with stabilising mutations and bound cyanopindolol
Class: receptor
Keywords: gpcr, membrane, receptor, palmitate, transducer, antagonist bound form, integral membrane protein, g-protein coupled receptor, g protein coupled receptor, thermostabilising point mutations, phosphoprotein, seven-helix receptor, lipoprotein, 7tm receptor, glycoprotein, transmembrane
Deposited on 2008-05-09, released 2008-06-24
The last revision prior to the SCOPe 2.08 freeze date was dated 2020-07-29, with a file datestamp of 2020-06-29.
Experiment type: XRAY
Resolution: 2.7 Å
R-factor: N/A
AEROSPACI score: 0.24 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: beta1 adrenergic receptor
    Species: MELEAGRIS GALLOPAVO [TaxId:9103]
    Database cross-references and differences (RAF-indexed):
    • PDB 2VT4
      • engineered mutation (37)
      • engineered mutation (59)
      • engineered mutation (85)
      • engineered mutation (196)
      • engineered mutation (266)
      • engineered mutation (277)
      • engineered mutation (297)
    • Uniprot P07700
    Domains in SCOPe 2.08: d2vt4a_
  • Chain 'B':
    Compound: beta1 adrenergic receptor
    Species: MELEAGRIS GALLOPAVO [TaxId:9103]
    Database cross-references and differences (RAF-indexed):
    • PDB 2VT4
      • engineered mutation (37)
      • engineered mutation (59)
      • engineered mutation (85)
      • engineered mutation (196)
      • engineered mutation (266)
      • engineered mutation (277)
      • engineered mutation (297)
    • Uniprot P07700
    Domains in SCOPe 2.08: d2vt4b_
  • Chain 'C':
    Compound: beta1 adrenergic receptor
    Species: MELEAGRIS GALLOPAVO [TaxId:9103]
    Database cross-references and differences (RAF-indexed):
    • PDB 2VT4
      • engineered mutation (37)
      • engineered mutation (59)
      • engineered mutation (85)
      • engineered mutation (196)
      • engineered mutation (266)
      • engineered mutation (277)
    • Uniprot P07700
    Domains in SCOPe 2.08: d2vt4c_
  • Chain 'D':
    Compound: beta1 adrenergic receptor
    Species: MELEAGRIS GALLOPAVO [TaxId:9103]
    Database cross-references and differences (RAF-indexed):
    • PDB 2VT4
      • engineered mutation (37)
      • engineered mutation (59)
      • engineered mutation (85)
      • engineered mutation (196)
      • engineered mutation (266)
      • engineered mutation (277)
    • Uniprot P07700
    Domains in SCOPe 2.08: d2vt4d_
  • Heterogens: P32, NA, SOG, D10, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >2vt4A (A:)
    mgaellsqqweagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvv
    gllvvpfgatlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryq
    slmtrarakviictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaia
    ssiisfyipllimifvalrvyreakeqirkidraskrkrvmlmrehkalktlgiimgvft
    lcwlpfflvnivnvfnrdlvpdwlfvafnwlgyansamnpiiycrspdfrkafkrllafp
    rkadrrlhhhhhh
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vt4A (A:)
    weagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvvgllvvpfga
    tlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryqslmtrarak
    viictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaiassiisfyip
    llimifvalrvyreakeqirehkalktlgiimgvftlcwlpfflvnivnvfnrdlvpdwl
    fvafnwlgyansamnpiiycrspdfrkafkrlla
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >2vt4B (B:)
    mgaellsqqweagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvv
    gllvvpfgatlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryq
    slmtrarakviictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaia
    ssiisfyipllimifvalrvyreakeqirkidraskrkrvmlmrehkalktlgiimgvft
    lcwlpfflvnivnvfnrdlvpdwlfvafnwlgyansamnpiiycrspdfrkafkrllafp
    rkadrrlhhhhhh
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vt4B (B:)
    qweagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvvgllvvpfg
    atlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryqslmtrara
    kviictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaiassiisfyi
    pllimifvalrvyreakeqirehkalktlgiimgvftlcwlpfflvnivnvfnrdlvpdw
    lfvafnwlgyansamnpiiycrspdfrkafkrllaf
    

  • Chain 'C':
    Sequence, based on SEQRES records: (download)
    >2vt4C (C:)
    mgaellsqqweagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvv
    gllvvpfgatlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryq
    slmtrarakviictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaia
    ssiisfyipllimifvalrvyreakeqirkidraskrkrvmlmrehkalktlgiimgvft
    lcwlpfflvnivnvfnrdlvpdwlfvafnwlgyansamnpiiycrspdfrkafkrllafp
    rkadrrlhhhhhh
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vt4C (C:)
    qweagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvvgllvvpfg
    atlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryqslmtrara
    kviictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaiassiisfyi
    pllimifvalrvyreakeqirehkalktlgiimgvftlcwlpfflvnivnvfnrdlvpdw
    lfvafnwlgyansamnpiiycrs
    

  • Chain 'D':
    Sequence, based on SEQRES records: (download)
    >2vt4D (D:)
    mgaellsqqweagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvv
    gllvvpfgatlvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryq
    slmtrarakviictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaia
    ssiisfyipllimifvalrvyreakeqirkidraskrkrvmlmrehkalktlgiimgvft
    lcwlpfflvnivnvfnrdlvpdwlfvafnwlgyansamnpiiycrspdfrkafkrllafp
    rkadrrlhhhhhh
    

    Sequence, based on observed residues (ATOM records): (download)
    >2vt4D (D:)
    eagmsllmalvvllivagnvlviaaigstqrlqtltnlfitslacadlvvgllvvpfgat
    lvvrgtwlwgsflcelwtsldvlcvtasietlcviaidrylaitspfryqslmtrarakv
    iictvwaisalvsflpimmhwwrdedpqalkcyqdpgccdfvtnrayaiassiisfyipl
    limifvalrvyreakeqirehkalktlgiimgvftlcwlpfflvnivnvfnrdlvpdwlf
    vafnwlgyansamnpiiycrspdfrkafkrll