PDB entry 2vo7
View 2vo7 on RCSB PDB site
Description: structure of pka complexed with 4-(4-chlorobenzyl)-1-(7h-pyrrolo(2,3-d)pyrimidin-4-yl)piperidin-4-ylamine
Class: transferase
Keywords: transferase, lipoprotein, ATP-binding, phosphoprotein, serine/threonine-protein kinase, nucleotide-binding, protein kinase inhibitor, camp, kinase, nucleus, myristate, cytoplasm
Deposited on
2008-02-08, released
2008-04-08
The last revision prior to the SCOP 1.75 freeze date was dated
2008-04-29, with a file datestamp of
2008-04-25.
Experiment type: XRAY
Resolution: 1.98 Å
R-factor: 0.19072
AEROSPACI score: 0.56
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-dependent protein kinase, alpha-catalytic subunit
Species: BOS TAURUS
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.75: d2vo7a1 - Chain 'I':
Compound: cAMP-dependent protein kinase inhibitor alpha
Database cross-references and differences (RAF-indexed):
- Heterogens: M05, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2vo7A (A:)
mgnaaaakkgseqesvkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvml
vkhmetgnhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymv
meyvpggemfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgy
iqvtdfgfakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppff
adqpiqiyekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfat
tdwiaiyqrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
Sequence, based on observed residues (ATOM records): (download)
>2vo7A (A:)
svkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvmlvkhmetgnhyamki
ldkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvmeyvpggemfshlr
rigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyiqvtdfgfakrvkg
rtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffadqpiqiyekivsg
kvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfattdwiaiyqrkveap
fipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
- Chain 'I':
No sequence available.