PDB entry 2uw9
View 2uw9 on RCSB PDB site
Description: structure of pkb-beta (akt2) complexed with 4-(4-chloro-phenyl)-4-(4-(1h-pyrazol-4-yl)-phenyl)-piperidine
Class: transferase/inhibitor complex
Keywords: transferase/inhibitor complex, wnt signaling pathway, serine/threonine-protein kinase, kinase, transferase, ATP-binding, phosphorylation, nucleotide-binding, alternative splicing, transferase/inhibitor complex
Deposited on
2007-03-19, released
2007-05-08
The last revision prior to the SCOP 1.75 freeze date was dated
2008-04-29, with a file datestamp of
2008-04-25.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.22585
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: rac-beta serine/threonine-protein kinase
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
- PDB 2UW9 (Start-341)
- Uniprot P31751 (5-End)
Domains in SCOP 1.75: d2uw9a1 - Chain 'C':
Compound: Glycogen synthase kinase-3 beta
Database cross-references and differences (RAF-indexed):
- Heterogens: GVP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2uw9A (A:)
gamdpkvtmndfdylkllgkgtfgkvilvrekatgryyamkilrkeviiakdevahtvte
srvlqntrhpfltalkyafqthdrlcfvmeyanggelffhlsrervfteerarfygaeiv
saleylhsrdvvyrdiklenlmldkdghikitdfglckegisdgatmktfcgtpeylape
vledndygravdwwglgvvmyemmcgrlpfynqdherlfelilmeeirfprtlspeaksl
lagllkkdpkqrlgggpsdakevmehrfflsinwqdvvqkkllppfkpqvtsevdtryfd
deftaqsititppdrydslglleldqreeqemfedfdyiadw
Sequence, based on observed residues (ATOM records): (download)
>2uw9A (A:)
kvtmndfdylkllgkgtfgkvilvrekatgryyamkilrkeviiakdevahtvtesrvlq
ntrhpfltalkyafqthdrlcfvmeyanggelffhlsrervfteerarfygaeivsaley
lhsrdvvyrdiklenlmldkdghikitdfglckegisdgatmktfcgtpeylapevledn
dygravdwwglgvvmyemmcgrlpfynqdherlfelilmeeirfprtlspeaksllagll
kkdpkqrlgggpsdakevmehrfflsinwqdvvqkkllppfkpqvtsevdtryfddefta
qsitqemfedfdyiadw
- Chain 'C':
No sequence available.