PDB entry 2rl5
View 2rl5 on RCSB PDB site
Description: Crystal structure of the VEGFR2 kinase domain in complex with a 2,3-dihydro-1,4-benzoxazine inhibitor
Class: transferase
Keywords: receptor tyrosine kinase, angiogenesis, , ATP-binding, Developmental protein, Differentiation, Glycoprotein, Host-virus interaction, Immunoglobulin domain, Membrane, Nucleotide-binding, Phosphorylation, Polymorphism, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2007-10-18, released
2008-04-08
The last revision prior to the SCOPe 2.07 freeze date was dated
2017-07-26, with a file datestamp of
2017-07-21.
Experiment type: XRAY
Resolution: 2.65 Å
R-factor: N/A
AEROSPACI score: 0.19
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Vascular endothelial growth factor receptor 2
Species: Homo sapiens [TaxId:9606]
Gene: KDR, FLK1
Database cross-references and differences (RAF-indexed):
- Uniprot P35968 (0-124)
- engineered (2)
- engineered (101)
- engineered (125)
- Uniprot P35968 (125-306)
Domains in SCOPe 2.07: d2rl5a1, d2rl5a2 - Heterogens: 2RL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2rl5A (A:)
ehaerlpydaskwefprdrlklgkplgrgafgqvieadafgidktatcrtvavkmlkega
thsehralmselkilihighhlnvvnllgactkpggplmvitefckfgnlstylrskrne
fvpykvapedlykdfltlehlicysfqvakgmeflasrkcihrdlaarnillseknvvki
cdfglardiykdpdyvrkgdarlplkwmapetifdrvytiqsdvwsfgvllweifslgas
pypgvkideefcrrlkegtrmrapdyttpemyqtmldcwhgepsqrptfselvehlgnll
qanaqqdrhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>2rl5A (A:)
ehaerlpydaskwefprdrlklgkplgrgqvieadafgidktatcrtvavkmlkegaths
ehralmselkilihighhlnvvnllgactkpggplmvitefckfgnlstylrskrnefvp
ykvapedlykdfltlehlicysfqvakgmeflasrkcihrdlaarnillseknvvkicdf
gldarlplkwmapetifdrvytiqsdvwsfgvllweifslgaspypgvkideefcrrlke
gtrmrapdyttpemyqtmldcwhgepsqrptfselvehlgnllqanaqqdrhhh