PDB entry 2r5q
View 2r5q on RCSB PDB site
Description: Crystal Structure Analysis of HIV-1 Subtype C Protease Complexed with Nelfinavir
Class: hydrolase
Keywords: HIV-1 subtype C, Aspartyl protease, Hydrolase, Protease, VIRAL PROTEIN
Deposited on
2007-09-04, released
2007-11-20
The last revision prior to the SCOPe 2.04 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.253
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q50CM2 (0-98)
- engineered (6)
- engineered (32)
- conflict (36)
- engineered (62)
Domains in SCOPe 2.04: d2r5qa_ - Chain 'B':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q50CM2 (0-98)
- engineered (6)
- engineered (32)
- conflict (36)
- engineered (62)
Domains in SCOPe 2.04: d2r5qb_ - Chain 'C':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q50CM2 (0-98)
- engineered (6)
- engineered (32)
- conflict (36)
- engineered (62)
Domains in SCOPe 2.04: d2r5qc_ - Chain 'D':
Compound: Protease
Species: Human immunodeficiency virus 1 [TaxId:11676]
Gene: pol
Database cross-references and differences (RAF-indexed):
- Uniprot Q50CM2 (0-98)
- engineered (6)
- engineered (32)
- conflict (36)
- engineered (62)
Domains in SCOPe 2.04: d2r5qd_ - Heterogens: 1UN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>2r5qA (A:)
pqitlwkrplvsikvggqikealldtgaddtvieeialpgrwkpkmiggiggfikvrqyd
qiiieicgkkaigtvlvgptpvniigrnmltqlgctlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>2r5qB (B:)
pqitlwkrplvsikvggqikealldtgaddtvieeialpgrwkpkmiggiggfikvrqyd
qiiieicgkkaigtvlvgptpvniigrnmltqlgctlnf
- Chain 'C':
Sequence; same for both SEQRES and ATOM records: (download)
>2r5qC (C:)
pqitlwkrplvsikvggqikealldtgaddtvieeialpgrwkpkmiggiggfikvrqyd
qiiieicgkkaigtvlvgptpvniigrnmltqlgctlnf
- Chain 'D':
Sequence; same for both SEQRES and ATOM records: (download)
>2r5qD (D:)
pqitlwkrplvsikvggqikealldtgaddtvieeialpgrwkpkmiggiggfikvrqyd
qiiieicgkkaigtvlvgptpvniigrnmltqlgctlnf