PDB entry 2qxs
View 2qxs on RCSB PDB site
Description: Crystal Structure of Antagonizing Mutant 536S of the Estrogen Receptor Alpha Ligand Binding Domain Complexed to Raloxifene
Class: transcription
Keywords: Protein-Ligand Complex, DNA-binding, Lipid-binding, Metal-binding, Nucleus, Phosphorylation, Receptor, Steroid-binding, Transcription, Transcription regulation, Zinc-finger
Deposited on
2007-08-12, released
2008-09-02
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-25, with a file datestamp of
2017-10-20.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: N/A
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Gene: ESR1, ESR, NR3A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2qxsa_ - Chain 'B':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Gene: ESR1, ESR, NR3A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2qxsb_ - Heterogens: RAL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2qxsA (A:)
sikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvh
minwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgk
cvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhih
rvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvps
ydlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>2qxsA (A:)
lalsltadqmvsalldaeppilyseydprpfsasmmglltnladrelvhminwakrvpgf
vdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmveifdm
llatssrfrmmnlqgeefvclksiillnsgvytftlksleekdhihrvldkitdtlihlm
akagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpsydlllemldah
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2qxsB (B:)
sikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvh
minwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgk
cvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhih
rvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvps
ydlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>2qxsB (B:)
lalsltadqmvsalldaeppilyseyasmmglltnladrelvhminwakrvpgfvdltlh
dqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmveifdmllatss
rfrmmnlqgeefvclksiillnsgvyleekdhihrvldkitdtlihlmakagltlqqqhq
rlaqlllilshirhmsnkgmehlysmkcknvvpsydlllemldahr