PDB entry 2qd8

View 2qd8 on RCSB PDB site
Description: HIV-1 Protease Mutant I84V with potent Antiviral inhibitor GRL-98065
Class: hydrolase
Keywords: HIV-1 protease mutant I84V, protease inhibitor, HYDROLASE
Deposited on 2007-06-20, released 2008-04-22
The last revision prior to the SCOP 1.75 freeze date was dated 2008-04-22, with a file datestamp of 2008-04-18.
Experiment type: XRAY
Resolution: 1.35 Å
R-factor: 0.133
AEROSPACI score: 0.9 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Protease
    Species: Human immunodeficiency virus type 1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P03367
      • engineered (6)
      • engineered (32)
      • engineered (62)
      • engineered (66)
      • engineered (83)
      • engineered (94)
    Domains in SCOP 1.75: d2qd8a1
  • Chain 'B':
    Compound: Protease
    Species: Human immunodeficiency virus type 1
    Database cross-references and differences (RAF-indexed):
    • Uniprot P03367 (0-98)
      • engineered (6)
      • engineered (32)
      • engineered (62)
      • engineered (66)
      • engineered (83)
      • engineered (94)
    Domains in SCOP 1.75: d2qd8b1
  • Heterogens: NA, CL, ACT, 065, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence; same for both SEQRES and ATOM records: (download)
    >2qd8A (A:)
    pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpkmiggiggfikvrqyd
    qiiieiaghkaigtvlvgptpvnvigrnlltqigatlnf
    

  • Chain 'B':
    Sequence; same for both SEQRES and ATOM records: (download)
    >2qd8B (B:)
    pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpkmiggiggfikvrqyd
    qiiieiaghkaigtvlvgptpvnvigrnlltqigatlnf