PDB entry 2qab
View 2qab on RCSB PDB site
Description: Crystal Structure of Estrogen Receptor Alpha Ligand Binding Domain Mutant 537S Complexed with an Ethyl Indazole Compound
Class: transcription
Keywords: Protein-Ligand Complex, TRANSCRIPTION
Deposited on
2007-06-14, released
2008-03-18
The last revision prior to the SCOPe 2.07 freeze date was dated
2017-10-18, with a file datestamp of
2017-10-13.
Experiment type: XRAY
Resolution: 1.89 Å
R-factor: N/A
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Gene: ESR1, ESR, NR3A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d2qaba_ - Chain 'B':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Gene: ESR1, ESR, NR3A1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d2qabb_ - Chain 'C':
Compound: nuclear receptor coactivator 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Chain 'D':
Compound: nuclear receptor coactivator 2
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: EI1, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2qabA (A:)
sikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvh
minwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgk
cvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhih
rvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpl
sdlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>2qabA (A:)
slalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrv
pgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmvei
fdmllatssrfrmmnlqgeefvclksiillnsgvytfeekdhihrvldkitdtlihlmak
agltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplsdlllemldahr
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2qabB (B:)
sikrskknslalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvh
minwakrvpgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgk
cvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhih
rvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpl
sdlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>2qabB (B:)
slalsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrv
pgfvdltlhdqvhllecawleilmiglvwrsmehpgkllfapnllldrnqgkcvegmvei
fdmllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitd
tlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvplsdllleml
dahrl
- Chain 'C':
No sequence available.
- Chain 'D':
No sequence available.