PDB entry 2pir
View 2pir on RCSB PDB site
Description: Androgen receptor LBD with small molecule
Class: hormone receptor
Keywords: androgen receptor coactivator binding inhibitors AF-2 pocket, HORMONE RECEPTOR
Deposited on
2007-04-13, released
2007-09-25
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-18, with a file datestamp of
2017-10-13.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: N/A
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Androgen receptor
Species: Homo sapiens [TaxId:9606]
Gene: AR, DHTR, NR3C4
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2pira_ - Heterogens: SO4, DHT, NK, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2pirA (A:)
cqpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnl
hvddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksrmysqcvrmr
hlsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrkn
ptscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkils
gkvkpiyfhtq
Sequence, based on observed residues (ATOM records): (download)
>2pirA (A:)
cqpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnl
hvddqmaviqyswmglmvfamgwrsftnvnsrmlyfapdlvfneyrmhksrmysqcvrmr
hlsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrkn
ptscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkils
gkvkpiyfht