PDB entry 2pe1
View 2pe1 on RCSB PDB site
Description: CRYSTAL STRUCTURE OF HUMAN PHOSPHOINOSITIDE-DEPENDENT PROTEIN KINASE 1 (PDK1) {2-Oxo-3-[1-(1H-pyrrol-2-yl)-eth-(Z)-ylidene]-2,3-dihydro-1H-indol-5-yl}-urea {BX-517} COMPLEX
Class: transferase
Keywords: protein inhibitor complex, serine kinase
Deposited on
2007-04-01, released
2007-06-12
The last revision prior to the SCOP 1.73 freeze date was dated
2007-07-17, with a file datestamp of
2007-07-13.
Experiment type: XRAY
Resolution: 2.14 Å
R-factor: 0.224
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide-dependent protein kinase 1
Species: HOMO SAPIENS
Gene: PDPK1, PDK1
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d2pe1a1 - Heterogens: SO4, 517, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2pe1A (A:)
prkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerdv
msrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsal
eylhgkgiihrdlkpenillnedmhiqitdfgtakvlspeskqaransfvgtaqyvspel
lteksackssdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlv
ekllvldatkrlgceemegygplkahpffesvtwenlhqqtppklt
Sequence, based on observed residues (ATOM records): (download)
>2pe1A (A:)
prkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerdv
msrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsal
eylhgkgiihrdlkpenillnedmhiqitdfgtakvlsfvgtaqyvspellteksackss
dlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvldatk
rlgceemegygplkahpffesvtwenlhqqtppklt