PDB entry 2pd5
View 2pd5 on RCSB PDB site
Description: Human aldose reductase mutant V47I complexed with zopolrestat
Class: oxidoreductase
Keywords: TIM barrel, V47I mutant, OXIDOREDUCTASE
Deposited on
2007-03-31, released
2008-04-01
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 1.6 Å
R-factor: 0.173
AEROSPACI score: 0.58
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: aldose reductase
Species: Homo sapiens [TaxId:9606]
Gene: ALR2
Database cross-references and differences (RAF-indexed):
- Uniprot P15121 (Start-315)
- conflict (4)
- engineered (47)
Domains in SCOPe 2.06: d2pd5a_ - Heterogens: NAP, ZST, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2pd5A (A:)
masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahiyqnenevgvaiq
eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwptgfkpgk
effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
llsctshkdypfheef
Sequence, based on observed residues (ATOM records): (download)
>2pd5A (A:)
asrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahiyqnenevgvaiqe
klreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwptgfkpgke
ffpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykpa
vnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaakh
nkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvcal
lsctshkdypfheef