PDB entry 2p2h
View 2p2h on RCSB PDB site
Description: Crystal structure of the VEGFR2 kinase domain in complex with a pyridinyl-triazine inhibitor
Class: Transferase
Keywords: receptor tyrosine kinase, KDR, Transferase
Deposited on
2007-03-07, released
2007-03-20
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: 0.205
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Vascular endothelial growth factor receptor 2
Species: Homo sapiens [TaxId:9606]
Gene: KDR, FLK1
Database cross-references and differences (RAF-indexed):
- Uniprot P35968 (0-124)
- engineered (2)
- engineered (101)
- engineered (125)
- cloning artifact (307)
- expression tag (308-310)
- Uniprot P35968 (125-306)
Domains in SCOPe 2.05: d2p2ha_ - Heterogens: 994, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2p2hA (A:)
ehaerlpydaskwefprdrlklgkplgrgafgqvieadafgidktatcrtvavkmlkega
thsehralmselkilihighhlnvvnllgactkpggplmvitefckfgnlstylrskrne
fvpykvapedlykdfltlehlicysfqvakgmeflasrkcihrdlaarnillseknvvki
cdfglardiykdpdyvrkgdarlplkwmapetifdrvytiqsdvwsfgvllweifslgas
pypgvkideefcrrlkegtrmrapdyttpemyqtmldcwhgepsqrptfselvehlgnll
qanaqqdrhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>2p2hA (A:)
ehaerlpydaskwefprdrlklgkplgrqvieadafgidktatcrtvavkmlkegathse
hralmselkilihighhlnvvnllgactkpggplmvitefckfgnlstylrskrnefvpy
kvapedlykdfltlehlicysfqvakgmeflasrkcihrdlaarnillseknvvkicdfg
larlplkwmapetifdrvytiqsdvwsfgvllweifslgaspypgvkideefcrrlkegt
rmrapdyttpemyqtmldcwhgepsqrptfselvehlgnllqanaqqdrhhh