PDB entry 2np8
View 2np8 on RCSB PDB site
Description: Structural Basis for the Inhibition of Aurora A Kinase by a Novel Class of High Affinity Disubstituted Pyrimidine Inhibitors
Class: Transferase
Keywords: Aurora A kinase, AIK, aurora 2 kinase, kinase, kinase inhibitor, Transferase
Deposited on
2006-10-26, released
2006-12-26
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-09-01, with a file datestamp of
2009-08-28.
Experiment type: XRAY
Resolution: 2.25 Å
R-factor: 0.246
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase 6
Species: Homo sapiens [TaxId:9606]
Gene: AIK
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d2np8a_ - Heterogens: SO4, CC3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2np8A (A:)
gamgskrqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlr
reveiqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyite
lanalsychskrvihrdikpenlllgsagelkiadfgwsvhapssrrttlcgtldylppe
miegrmhdekvdlwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardl
isrllkhnpsqrpmlrevlehpwitansskps
Sequence, based on observed residues (ATOM records): (download)
>2np8A (A:)
qwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrreveiqs
hlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitelanalsy
chskrvihrdikpenlllgsagelkiadfgwsvhapssrtldylppemiegrmhdekvdl
wslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardlisrllkhnpsqrp
mlrevlehpwitanss