PDB entry 2jkk
View 2jkk on RCSB PDB site
Description: focal adhesion kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor
Class: transferase
Keywords: tyrosine-protein kinase, tyrosine- protein kinase, kinase, membrane, transferase, ATP-binding, integrin signaling, nucleotide-binding, focal adhesion, cell migration, kinase inhibitor, cell junction, cell membrane, phosphoprotein
Deposited on
2008-08-28, released
2008-09-09
The last revision prior to the SCOPe 2.01 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-31.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.18189
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Focal adhesion kinase 1
Species: Gallus gallus [TaxId:9031]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d2jkka_ - Heterogens: SO4, BI9, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2jkkA (A:)
strdyeiqrerielgrcigegqfgdvhqgiymspenpamavaiktcknctsdsvrekflq
ealtmrqfdhphivkligvitenpvwiimelctlgelrsflqvrkfsldlaslilyayql
stalayleskrfvhrdiaarnvlvsatdcvklgdfglsrymedstyykaskgklpikwma
pesinfrrftsasdvwmfgvcmweilmhgvkpfqgvknndvigriengerlpmppncppt
lyslmtkcwaydpsrrprftelkaqlstileeeklq
Sequence, based on observed residues (ATOM records): (download)
>2jkkA (A:)
rdyeiqrerielgrcigegqfgdvhqgiymspenpamavaiktcknctsdsvrekflqea
ltmrqfdhphivkligvitenpvwiimelctlgelrsflqvrkfsldlaslilyayqlst
alayleskrfvhrdiaarnvlvsatdcvklgdfglsrlpikwmapesinfrrftsasdvw
mfgvcmweilmhgvkpfqgvknndvigriengerlpmppncpptlyslmtkcwaydpsrr
prftelkaqlstileeek