PDB entry 2i1m
View 2i1m on RCSB PDB site
Description: cFMS tyrosine kinase (tie2 KID) in complex with an arylamide inhibitor
Class: transferase
Keywords: Kinase Domain, Kinase Inhibitor Complex, transferase
Deposited on
2006-08-14, released
2006-11-28
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.25
AEROSPACI score: 0.44
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Macrophage colony-stimulating factor 1 receptor
Species: Homo sapiens [TaxId:9606]
Gene: CSF1R
Database cross-references and differences (RAF-indexed):
- Uniprot P07333 (Start-143)
- see remark 999 (144-150)
- see remark 999 (158-162)
- Uniprot P07333 (163-End)
Domains in SCOPe 2.01: d2i1ma_ - Heterogens: 5CN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2i1mA (A:)
gvdykykqkpkyqvrwkiiesyegnsytfidptqlpynekwefprnnlqfgktlgagafg
kvveatafglgkedavlkvavkmlkstahadekealmselkimshlgqhenivnllgact
hggpvlviteyccygdllnflrrksrvletdpafaianstastrdllhfssqvaqgmafl
askncihrdvaarnvlltnghvakigdfglardimndsnyivkgnarlpvkwmapesifd
cvytvqsdvwsygillweifslglnpypgilvnskfyklvkdgyqmaqpafapkniysim
qacwalepthrptfqqicsflqeqaqedrrerd
Sequence, based on observed residues (ATOM records): (download)
>2i1mA (A:)
qvrwkiiesynsytfidptqlpynekwefprnnlqfgktlgagafgkvveatafglgked
avlkvavkmlkstahadekealmselkimshlgqhenivnllgacthggpvlviteyccy
gdllnflrrksrvletdstastrdllhfssqvaqgmaflaskncihrdvaarnvlltngh
vakigdfglardimndsnyivkgnarlpvkwmapesifdcvytvqsdvwsygillweifs
lglnpypgilvnskfyklvkdgyqmaqpafapkniysimqacwalepthrptfqqicsfl
qeqaqedrrer