PDB entry 2hy8
View 2hy8 on RCSB PDB site
Description: PAK1 complex with ST2001
Class: transferase
Keywords: Typical fold of Ser/Thr kinases. Inhibitor is bound between the N-terminal and C-terminal domains., TRANSFERASE
Deposited on
2006-08-04, released
2006-11-07
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-11, with a file datestamp of
2017-10-06.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain '1':
Compound: Serine/threonine-protein kinase PAK 1
Species: Homo sapiens [TaxId:9606]
Gene: PAK1
Database cross-references and differences (RAF-indexed):
- Uniprot Q13153 (0-End)
- engineered (50)
- engineered (174)
- conflict (254)
Domains in SCOPe 2.08: d2hy81_ - Heterogens: 1ST, HOH
PDB Chain Sequences:
- Chain '1':
Sequence, based on SEQRES records: (download)
>2hy81 (1:)
sdeeileklrsivsvgdpkkkytrfekigqgasgtvytamdvatgqevairqmnlqqqpk
keliineilvmrenknpnivnyldsylvgdelwvvmeylaggsltdvvtetcmdegqiaa
vcreclqaleflhsnqvihrdiksdnillgmdgsvkltdfgfcaqitpeqskrsemvgtp
ywmapevvtrkaygpkvdiwslgimaiemiegeppylnenplralyliatngtpelqnpe
klsaifrdflnrcldmdvekrgsakellqhqflkiakplssltpliaaakeatknnh
Sequence, based on observed residues (ATOM records): (download)
>2hy81 (1:)
sdeeileklrsivsvgdpkkkytrfekigqgasgtvytamdvatgqevairqmnlqqqpk
keliineilvmrenknpnivnyldsylvgdelwvvmeylaggsltdvvtetcmdegqiaa
vcreclqaleflhsnqvihrdiksdnillgmdgsvkltdfgfcaqitpeqskrsemvgtp
ywmapevvtrkaygpkvdiwslgimaiemiegeppylnenplralyliatngtpelqnpe
klsaifrdflnrcldmdvekrgsakellqhqflkiakplssltpliaaakeat