PDB entry 2hy8

View 2hy8 on RCSB PDB site
Description: PAK1 complex with ST2001
Class: transferase
Keywords: Typical fold of Ser/Thr kinases. Inhibitor is bound between the N-terminal and C-terminal domains., TRANSFERASE
Deposited on 2006-08-04, released 2006-11-07
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-10-11, with a file datestamp of 2017-10-06.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31 (click here for full SPACI score report)

Chains and heterogens:

  • Chain '1':
    Compound: Serine/threonine-protein kinase PAK 1
    Species: Homo sapiens [TaxId:9606]
    Gene: PAK1
    Database cross-references and differences (RAF-indexed):
    • Uniprot Q13153 (0-End)
      • engineered (50)
      • engineered (174)
      • conflict (254)
    Domains in SCOPe 2.08: d2hy81_
  • Heterogens: 1ST, HOH

PDB Chain Sequences:

  • Chain '1':
    Sequence, based on SEQRES records: (download)
    >2hy81 (1:)
    sdeeileklrsivsvgdpkkkytrfekigqgasgtvytamdvatgqevairqmnlqqqpk
    keliineilvmrenknpnivnyldsylvgdelwvvmeylaggsltdvvtetcmdegqiaa
    vcreclqaleflhsnqvihrdiksdnillgmdgsvkltdfgfcaqitpeqskrsemvgtp
    ywmapevvtrkaygpkvdiwslgimaiemiegeppylnenplralyliatngtpelqnpe
    klsaifrdflnrcldmdvekrgsakellqhqflkiakplssltpliaaakeatknnh
    

    Sequence, based on observed residues (ATOM records): (download)
    >2hy81 (1:)
    sdeeileklrsivsvgdpkkkytrfekigqgasgtvytamdvatgqevairqmnlqqqpk
    keliineilvmrenknpnivnyldsylvgdelwvvmeylaggsltdvvtetcmdegqiaa
    vcreclqaleflhsnqvihrdiksdnillgmdgsvkltdfgfcaqitpeqskrsemvgtp
    ywmapevvtrkaygpkvdiwslgimaiemiegeppylnenplralyliatngtpelqnpe
    klsaifrdflnrcldmdvekrgsakellqhqflkiakplssltpliaaakeat