PDB entry 2h6g
View 2h6g on RCSB PDB site
Description: W102T Protein Farnesyltransferase Mutant Complexed with a Geranylgeranylated DDPTASACVLS Peptide Product at 1.85A Resolution
Class: transferase
Keywords: FTase, farnesyltransferase, farnesyl transferase, prenyltransferase, CaaX, Ras, lipid modification, prenylation, substrate selectivity, transferase
Deposited on
2006-05-31, released
2006-08-29
The last revision prior to the SCOPe 2.03 freeze date was dated
2010-10-13, with a file datestamp of
2010-10-08.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.187
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Protein farnesyltransferase/geranylgeranyltransferase type I alpha subunit
Species: Homo sapiens [TaxId:9606]
Gene: Human FTase alpha subunit
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d2h6ga1 - Chain 'B':
Compound: Protein farnesyltransferase beta subunit
Species: Homo sapiens [TaxId:9606]
Gene: Human FTase beta subunit
Database cross-references and differences (RAF-indexed):
- Chain 'P':
Compound: farnesylated peptide
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: SUC, ZN, GER, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2h6gA (A:)
maategvgeaaqggepgqpaqpppqphppppqqqhkeemaaeageavaspmddgfvslds
psyvlyrdraewadidpvpqndgpnpvvqiiysdkfrdvydyfravlqrderserafklt
rdaielnaanytvwhfrrvllkslqkdlheemnyitaiieeqpknyqvwhhrrvlvewlr
dpsqelefiadilnqdaknyhawqhrqwviqefklwdnelqyvdqllkedvrnnsvwnqr
yfvisnttgyndravlerevqytlemiklvphnesawnylkgilqdrglskypnllnqll
dlqpshsspyliaflvdiyedmlenqcdnkedilnkalelceilakekdtirkeywryig
rslqskhstendsptnvqqeef
Sequence, based on observed residues (ATOM records): (download)
>2h6gA (A:)
fvsldspsyvlyrdraewadidpvpqndgpnpvvqiiysdkfrdvydyfravlqrderse
rafkltrdaielnaanytvwhfrrvllkslqkdlheemnyitaiieeqpknyqvwhhrrv
lvewlrdpsqelefiadilnqdaknyhawqhrqwviqefklwdnelqyvdqllkedvrnn
svwnqryfvisnttgyndravlerevqytlemiklvphnesawnylkgilqdrglskypn
llnqlldlqpshsspyliaflvdiyedmlenqcdnkedilnkalelceilakekdtirke
ywryigrslqskhst
- Chain 'B':
No sequence available.
- Chain 'P':
No sequence available.