PDB entry 2gnj
View 2gnj on RCSB PDB site
Description: PKA three fold mutant model of Rho-kinase with Y-27632
Class: transferase/transferase inhibitor
Keywords: PKA, surrogate, Rho-kinase, H1152P, inhibitor, TRANSFERASE/TRANSFERASE INHIBITOR COMPLEX
Deposited on
2006-04-10, released
2006-05-23
The last revision prior to the SCOPe 2.01 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.28 Å
R-factor: 0.19
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-dependent protein kinase, alpha-catalytic subunit
Species: Bos taurus [TaxId:9913]
Gene: PRKACA
Database cross-references and differences (RAF-indexed):
- Uniprot P00517 (Start-349)
- engineered (48)
- engineered (180)
- engineered (182)
- modified residue (196)
- modified residue (337)
Domains in SCOPe 2.01: d2gnja_ - Chain 'I':
Compound: cAMP-dependent protein kinase inhibitor alpha
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: Y27, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2gnjA (A:)
gnaaaakkgseqesvkeflakakedflkkwenpaqntahldqferiktigtgsfgrvmlv
khmetgnhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvm
eyvpggemfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyi
kvadfgfakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffa
dqpiqiyekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfatt
dwiaiyqrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
Sequence, based on observed residues (ATOM records): (download)
>2gnjA (A:)
svkeflakakedflkkwenpaqntahldqferiktigtgsfgrvmlvkhmetgnhyamki
ldkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvmeyvpggemfshlr
rigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyikvadfgfakrvkg
rtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffadqpiqiyekivsg
kvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfattdwiaiyqrkveap
fipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
- Chain 'I':
No sequence available.