PDB entry 2fyp
View 2fyp on RCSB PDB site
Description: GRP94 in complex with the novel HSP90 Inhibitor Radester amine
Class: chaperone
Keywords: GRP94, HSP82, HSP90, HTPG, chaperone, ligand, radicicol, geldanamycin, radester, radamide
Deposited on
2006-02-08, released
2007-02-06
The last revision prior to the SCOPe 2.07 freeze date was dated
2017-08-02, with a file datestamp of
2017-07-28.
Experiment type: XRAY
Resolution: 1.95 Å
R-factor: N/A
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Endoplasmin
Species: Canis lupus [TaxId:9615]
Gene: TRA1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d2fypa2, d2fypa3 - Chain 'B':
Compound: Endoplasmin
Species: Canis lupus [TaxId:9615]
Gene: TRA1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d2fypb2, d2fypb3 - Heterogens: RDE, PG4, 1PE, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2fypA (A:)
gshmlreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltden
alagneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqed
gqstseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrg
ttitlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktggggktvwdwelmn
Sequence, based on observed residues (ATOM records): (download)
>2fypA (A:)
gshmlreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltden
alagneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqed
gqstseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrg
ttitlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktktvwdwelmn
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2fypB (B:)
gshmlreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltden
alagneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqed
gqstseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrg
ttitlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktggggktvwdwelmn
Sequence, based on observed residues (ATOM records): (download)
>2fypB (B:)
gshmlreksekfafqaevnrmmkliinslyknkeiflrelisnasdaldkirlisltden
alagneeltvkikcdkeknllhvtdtgvgmtreelvknlgtiaksgtseflnkmteaqed
gqstseligqfgvgfysaflvadkvivtskhnndtqhiwesdsnefsviadprgntlgrg
ttitlvlkeeasdyleldtiknlvkkysqfinfpiyvwssktktvwdwelmn