PDB entry 2f8c
View 2f8c on RCSB PDB site
Description: Crystal structure of FPPS in complex with Zoledronate
Class: transferase
Keywords: Mevalonate pathway, ; isoprene biosynthesis; cholesterol biosynthesis; bisphosphonate inhibitor, TRANSFERASE
Deposited on
2005-12-02, released
2006-02-28
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-18, with a file datestamp of
2017-10-13.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: N/A
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'F':
Compound: Farnesyl Diphosphate Synthase
Species: Homo sapiens [TaxId:9606]
Gene: FDPS, FPS, KIAA1293
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2f8cf_ - Heterogens: PO4, MG, ZOL, HOH
PDB Chain Sequences:
- Chain 'F':
Sequence, based on SEQRES records: (download)
>2f8cF (F:)
gpnsdvyaqekqdfvqhfsqivrvltedemghpeigdaiarlkevleynaiggkynrglt
vvvafrelveprkqdadslqrawtvgwcvellqafflvaddimdssltrrgqicwyqkpg
vgldaindanlleaciyrllklycreqpyylnlielflqssyqteigqtldlltapqgnv
dlvrftekryksivkyktafysfylpiaaamymagidgekehanakkillemgeffqiqd
dyldlfgdpsvtgkigtdiqdnkcswlvvqclqratpeqyqilkenygqkeaekvarvka
lyeeldlpavflqyeedsyshimalieqyaaplppavflglarkiykrrk
Sequence, based on observed residues (ATOM records): (download)
>2f8cF (F:)
dvyaqekqdfvqhfsqivrvltedemghpeigdaiarlkevleynaiggkynrgltvvva
frelveprkqdadslqrawtvgwcvellqafflvaddimdssltrrgqicwyqkpgvgld
aindanlleaciyrllklycreqpyylnlielflqssyqteigqtldlltapqgnvdlvr
ftekryksivkyktafysfylpiaaamymagidgekehanakkillemgeffqiqddyld
lfgdpsvtgkigtdiqdnkcswlvvqclqratpeqyqilkenygqkeaekvarvkalyee
ldlpavflqyeedsyshimalieqyaaplppavflglarkiyk