PDB entry 2f7z
View 2f7z on RCSB PDB site
Description: Protein Kinase A bound to (R)-1-(1H-Indol-3-ylmethyl)-2-(2-pyridin-4-yl-[1,7]naphtyridin-5-yloxy)-ehylamine
Class: transferase
Keywords: Protein Kinase A, AKT inhibitors, TRANSFERASE
Deposited on
2005-12-01, released
2006-06-27
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 3 Å
R-factor: 0.246
AEROSPACI score: 0.19
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'E':
Compound: cAMP-dependent protein kinase, alpha-catalytic subunit
Species: Bos taurus [TaxId:9913]
Gene: PRKACA
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d2f7ze_ - Chain 'I':
Compound: PKI, inhibitory peptide
Database cross-references and differences (RAF-indexed):
- Heterogens: 6EA
PDB Chain Sequences:
- Chain 'E':
Sequence, based on SEQRES records: (download)
>2f7zE (E:)
mgnaaaakkgseqesvkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvml
vkhmetgnhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymv
meyvpggemfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgy
iqvtdfgfakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppff
adqpiqiyekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfat
tdwiaiyqrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
Sequence, based on observed residues (ATOM records): (download)
>2f7zE (E:)
vkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvmlvkhmetgnhyamkil
dkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvmeyvpggemfshlrr
igrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyiqvtdfgfakrvkgr
twtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffadqpiqiyekivsgk
vrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfattdwiaiyqrkveapf
ipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
- Chain 'I':
No sequence available.