PDB entry 2f2c
View 2f2c on RCSB PDB site
Description: X-ray structure of human CDK6-Vcyclinwith the inhibitor aminopurvalanol
Class: cell cycle/transferase
Keywords: Small molecule inhibitor bound between N-terminal and C-terminal domain of kinase, CELL CYCLE-TRANSFERASE COMPLEX
Deposited on
2005-11-16, released
2006-06-13
The last revision prior to the SCOPe 2.07 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: 0.241
AEROSPACI score: 0.22
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cyclin homolog
Species: Herpesvirus saimiri (strain 11) [TaxId:10383]
Gene: 72, ECLF2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d2f2ca1, d2f2ca2 - Chain 'B':
Compound: cell division protein kinase 6
Species: Homo sapiens [TaxId:9606]
Gene: CDK6
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d2f2cb_ - Heterogens: SO4, AP9, DMS
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2f2cA (A:)
madspnrlnrakidsttmkdprvlnnlklrelllpkftslweiqtevtvdnrtilltwmh
llcesfeldksvfplsvsildrylckkqgtkktlqkigaacvligskirtvkpmtvsklt
ylscdcftnlelinqekdilealkwdteavlatdfliplcnalkipedlwpqlyeaastt
ickaliqpniallspglicaggllttietdntncrpwtcyledlssilnfstntvrtvkd
qvseafslydleil
Sequence, based on observed residues (ATOM records): (download)
>2f2cA (A:)
lnrakidsttmkdprvlnnlklrelllpkftslweiqtevtvdnrtilltwmhllcesfe
ldksvfplsvsildrylckkqgtkktlqkigaacvligskirtvkpmtvskltylsftnl
elinqekdilealkwdteavlatdfliplcnalkipedlwpqlyeaasttickaliqpni
allspglicaggllttietdntncrpwtcyledlssilnfstntvrtvkdqvseafslyd
leil
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2f2cB (B:)
mekdglcradqqyecvaeigegaygkvfkardlknggrfvalkrvrvqtgeegmplstir
evavlrhletfehpnvvrlfdvctvsrtdretkltlvfehvdqdlttyldkvpepgvpte
tikdmmfqllrgldflhshrvvhrdlkpqnilvtssgqikladfglariysfqmaltsvv
vtlwyrapevllqssyatpvdlwsvgcifaemfrrkplfrgssdvdqlgkildviglpge
edwprdvalprqafhsksaqpiekfvtdidelgkdlllkcltfnpakrisaysalshpyf
qdlercke
Sequence, based on observed residues (ATOM records): (download)
>2f2cB (B:)
adqqyecaeiggkvfkardlknggrfvalkrvrvqtgeegmplstirevavlrhletfeh
pnvvrlfdvctvstdretkltlvfehvdqdlttyldkvpepgvptetikdmmfqllrgld
flhshrvvhrdlkpqnilvtssgqikladfglariysfqmaltsvvvtlwyrapevllqs
syatpvdlwsvgcifaemfrrkplfrgssdvdqlgkildviglpgeedwpqafaqpiekf
vtdidelgkdlllkcltfnpakrisaysalshpyfqdler