PDB entry 2bgd
View 2bgd on RCSB PDB site
Description: structure-based design of protein tyrosine phosphatase-1b inhibitors
Class: hydrolase
Keywords: protein tyrosine phosphatase, 1, 2, 5-thiadiazolidin-3-one-1, 1-dioxide template, hydrolase
Deposited on
2004-12-21, released
2005-05-04
The last revision prior to the SCOPe 2.01 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-31.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.166
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: protein-tyrosine phosphatase non-receptor type 1
Species: HOMO SAPIENS
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.01: d2bgda1 - Heterogens: T1D, CL, PO4, NA, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2bgdA (A:)
memekefeqidksgswaaiyqdirheasdfpcrvaklpknknrnryrdvspfdhsriklh
qedndyinaslikmeeaqrsyiltqgplpntcghfwemvweqksrgvvmlnrvmekgslk
caqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfhyttwp
dfgvpespasflnflfkvresgslspehgpvvvhcsagigrsgtfcladtclllmdkrkd
pssvdikkvllemrkfrmgliqtadqlrfsylaviegakfimgdssvqdqwkelshedle
pppehipppprppkrilephn
Sequence, based on observed residues (ATOM records): (download)
>2bgdA (A:)
memekefeqidksgswaaiyqdirheasdfpcrvaklpknknrnryrdvspfdhsriklh
ndyinaslikmeeaqrsyiltqgplpntcghfwemvweqksrgvvmlnrvmekgslkcaq
ywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfhyttwpdfg
vpespasflnflfkvresgslspehgpvvvhcsagigrsgtfcladtclllmdkrkdpss
vdikkvllemrkfrmgliqtadqlrfsylaviegakfimgdssvqdqwkelshed