PDB entry 2bed
View 2bed on RCSB PDB site
Description: Structure of FPT bound to inhibitor SCH207736
Class: transferase
Keywords: FPT, PTase, Farnesyl, drug design, TRANSFERASE
Deposited on
2005-10-24, released
2006-08-08
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-01-24, with a file datestamp of
2018-01-19.
Experiment type: XRAY
Resolution: 2.7 Å
R-factor: N/A
AEROSPACI score: 0.19
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Protein farnesyltransferase/geranylgeranyltransferase type I alpha subunit
Species: Rattus norvegicus [TaxId:10116]
Gene: Fnta
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2beda_ - Chain 'B':
Compound: Protein farnesyltransferase beta subunit
Species: Rattus norvegicus [TaxId:10116]
Gene: Fntb
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d2bedb_ - Heterogens: ZN, FPP, 736, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>2bedA (A:)
gflsldsptyvlyrdraewadidpvpqndgpspvvqiiysekfrdvydyfravlqrders
erafkltrdaielnaanytvwhfrrvllrslqkdlqeemnyitaiieeqpknyqvwhhrr
vlvewlkdpsqelefiadilnqdaknyhawqhrqwviqefrlwdnelqyvdqllkedvrn
nsvwnqrhfvisnttgysdravlerevqytlemiklvphnesawnylkgilqdrglsryp
nllnqlldlqpshsspyliaflvdiyedmlenqcdnkedilnkalelceilakekdtirk
eywryigrslqsk
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>2bedB (B:)
lyslrpeharerlqddsvetvtsieqakveekiqevfssykfnhlvprlvlqrekhfhyl
krglrqltdayecldasrpwlcywilhslelldepipqivatdvcqflelcqspdggfgg
gpgqyphlaptyaavnalciigteeaynvinrekllqylyslkqpdgsflmhvggevdvr
saycaasvasltniitpdlfegtaewiarcqnweggiggvpgmeahggytfcglaalvil
kkerslnlksllqwvtsrqmrfeggfqgrcnklvdgcysfwqagllpllhralhaqgdpa
lsmshwmfhqqalqeyilmccqcpagglldkpgksrdfyhtcyclsglsiaqhfgsgaml
hdvvmgvpenvlqpthpvynigpdkviqatthflqkpvpgf