PDB entry 2ayp
View 2ayp on RCSB PDB site
Description: Crystal Structure of CHK1 with an Indol Inhibitor
Class: transferase
Keywords: Protein-Inhibitor Complex
Deposited on
2005-09-07, released
2006-09-12
The last revision prior to the SCOP 1.73 freeze date was dated
2006-09-12, with a file datestamp of
2007-06-04.
Experiment type: XRAY
Resolution: 2.9 Å
R-factor: 0.209
AEROSPACI score: 0.22
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: HOMO SAPIENS
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOP 1.73: d2aypa1 - Heterogens: 43A
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2aypA (A:)
mavpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicink
mlnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvy
lhgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellk
rrefhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsapla
llhkilvenpsaritipdikkdrwynkpl
Sequence, based on observed residues (ATOM records): (download)
>2aypA (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkpl