PDB entry 1wok
View 1wok on RCSB PDB site
Description: Crystal structure of catalytic domain of human poly(ADP-ribose) polymerase complexed with a quinoxaline-type inhibitor
Class: transferase
Keywords: protein-inhibitor complex, transferase
Deposited on
2004-08-20, released
2005-03-15
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-11, with a file datestamp of
2017-10-06.
Experiment type: XRAY
Resolution: 3 Å
R-factor: N/A
AEROSPACI score: 0.12
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Poly [ADP-ribose] polymerase-1
Species: Homo sapiens [TaxId:9606]
Gene: PPOL
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1woka1, d1woka2 - Chain 'B':
Compound: Poly [ADP-ribose] polymerase-1
Species: Homo sapiens [TaxId:9606]
Gene: PPOL
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1wokb1, d1wokb2 - Chain 'C':
Compound: Poly [ADP-ribose] polymerase-1
Species: Homo sapiens [TaxId:9606]
Gene: PPOL
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1wokc1, d1wokc2 - Chain 'D':
Compound: Poly [ADP-ribose] polymerase-1
Species: Homo sapiens [TaxId:9606]
Gene: PPOL
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d1wokd1, d1wokd2 - Heterogens: CNQ
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>1wokA (A:)
ksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysilsevqqavs
qgssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldievaysllrgg
sddsskdpidvnyeklktdikvvdrdseeaeiirkyvknthatthnaydlevidifkier
egecqrykpfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfgkgiyfadmv
sksanychtsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglgkttpdpsan
isldgvdvplgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkt
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>1wokB (B:)
ksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysilsevqqavs
qgssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldievaysllrgg
sddsskdpidvnyeklktdikvvdrdseeaeiirkyvknthatthnaydlevidifkier
egecqrykpfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfgkgiyfadmv
sksanychtsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglgkttpdpsan
isldgvdvplgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkt
- Chain 'C':
Sequence; same for both SEQRES and ATOM records: (download)
>1wokC (C:)
ksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysilsevqqavs
qgssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldievaysllrgg
sddsskdpidvnyeklktdikvvdrdseeaeiirkyvknthatthnaydlevidifkier
egecqrykpfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfgkgiyfadmv
sksanychtsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglgkttpdpsan
isldgvdvplgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkt
- Chain 'D':
Sequence; same for both SEQRES and ATOM records: (download)
>1wokD (D:)
ksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysilsevqqavs
qgssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldievaysllrgg
sddsskdpidvnyeklktdikvvdrdseeaeiirkyvknthatthnaydlevidifkier
egecqrykpfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfgkgiyfadmv
sksanychtsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglgkttpdpsan
isldgvdvplgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkt