PDB entry 1w2h
View 1w2h on RCSB PDB site
Description: crystal structure of mycobacterium tuberculosis thymidylate kinase complexed with azidothymidine monophosphate (azt-mp) (2.0 a resolution)
Class: transferase
Keywords: transferase, mycobacterium tuberculosis, thymidylate kinase, azt, inhibition mechanism, crystal structure
Deposited on
2004-07-06, released
2005-01-12
The last revision prior to the SCOPe 2.02 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.259
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: thymidylate kinase tmk
Species: Mycobacterium tuberculosis [TaxId:1773]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d1w2ha_ - Chain 'B':
Compound: thymidylate kinase tmk
Species: Mycobacterium tuberculosis [TaxId:1773]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d1w2hb_ - Heterogens: ATM, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1w2hA (A:)
mliaiegvdgagkrtlveklsgafraagrsvatlafprygqsvaadiaaealhgehgdla
ssvyamatlfaldragavhtiqglcrgydvvildryvasnaaysaarlhenaagkaaawv
qriefarlglpkpdwqvllavsaelagersrgraqrdpgrardnyerdaelqqrtgavya
elaaqgwggrwlvvgadvdpgrlaatlappdvps
Sequence, based on observed residues (ATOM records): (download)
>1w2hA (A:)
mliaiegvdgagkrtlveklsgafraagrsvatlafprygqsvaadiaaealhgehgdla
ssvyamatlfaldragavhtiqglcrgydvvildryvasnaaysaarlhenaagkaaawv
qriefarlglpkpdwqvllavsaelagerdaelqqrtgavyaelaaqgwggrwlvvgadv
dpgrlaatlap
- Chain 'B':
Sequence, based on SEQRES records: (download)
>1w2hB (B:)
mliaiegvdgagkrtlveklsgafraagrsvatlafprygqsvaadiaaealhgehgdla
ssvyamatlfaldragavhtiqglcrgydvvildryvasnaaysaarlhenaagkaaawv
qriefarlglpkpdwqvllavsaelagersrgraqrdpgrardnyerdaelqqrtgavya
elaaqgwggrwlvvgadvdpgrlaatlappdvps
Sequence, based on observed residues (ATOM records): (download)
>1w2hB (B:)
mliaiegvdgagkrtlveklsgafraagrsvatlafprygqsvaadiaaealhgehgdla
ssvyamatlfaldragavhtiqglcrgydvvildryvasnaaysaarlhenaagkaaawv
qriefarlglpkpdwqvllavsaelagersrgardnyerdaelqqrtgavyaelaaqgwg
grwlvvgadvdpgrlaatlap