PDB entry 1uu7
View 1uu7 on RCSB PDB site
Description: structure of human pdk1 kinase domain in complex with bim-2
Class: transferase
Keywords: protein kinase, pkb, pdk1, inhibitor, ly333531, bisindolyl maleimide, bim-1, diabetes, cancer, transferase, serine/threonine-protein kinase
Deposited on
2003-12-16, released
2004-03-04
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-31.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.235
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide dependent protein kinase-1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d1uu7a_ - Heterogens: GOL, BI2, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1uu7A (A:)
mdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsreyai
kilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngellky
irkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgtakvl
speskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragneyli
fqkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtwenl
hqqtppklta
Sequence, based on observed residues (ATOM records): (download)
>1uu7A (A:)
qprkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerd
vmsrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsa
leylhgkgiihrdlkpenillnedmhiqitdfgtakvlspransfvgtaqyvspelltek
sackssdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekll
vldatkrlgceemegygplkahpffesvtwenlhqqtppklt