PDB entry 1sve
View 1sve on RCSB PDB site
Description: Crystal Structure of Protein Kinase A in Complex with Azepane Derivative 1
Class: transferase
Keywords: kinase-inhibitor-complex, serine/threonine-protein kinase, balanol derivative, transferase
Deposited on
2004-03-29, released
2005-03-29
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 2.49 Å
R-factor: 0.202
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-dependent protein kinase, alpha-catalytic subunit
Species: Bos taurus [TaxId:9913]
Gene: PRKACA
Database cross-references and differences (RAF-indexed):
- Uniprot P00517 (Start-349)
- modified residue (9)
- modified residue (196)
- modified residue (337)
Domains in SCOPe 2.08: d1svea_ - Chain 'B':
Compound: cAMP-dependent protein kinase inhibitor, alpha form
Species: synthetic, synthetic
Database cross-references and differences (RAF-indexed):
- Heterogens: NA, I01, MG8, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>1sveA (A:)
gnaaaakkgseqesvkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvmlv
khmetgnhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvm
eyvpggemfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyi
qvtdfgfakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffa
dqpiqiyekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfatt
dwiaiyqrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
Sequence, based on observed residues (ATOM records): (download)
>1sveA (A:)
kkgseqesvkeflakakedflkkwenpaqntahldqferiktlgtgsfgrvmlvkhmetg
nhyamkildkqkvvklkqiehtlnekrilqavnfpflvklefsfkdnsnlymvmeyvpgg
emfshlrrigrfsepharfyaaqivltfeylhsldliyrdlkpenllidqqgyiqvtdfg
fakrvkgrtwtlcgtpeylapeiilskgynkavdwwalgvliyemaagyppffadqpiqi
yekivsgkvrfpshfssdlkdllrnllqvdltkrfgnlkngvndiknhkwfattdwiaiy
qrkveapfipkfkgpgdtsnfddyeeeeirvsinekcgkefsef
- Chain 'B':
No sequence available.